SCHEMBL5723934

SCHEMBL5723934

NC(=O)c1ccccc1Cc1ccc(O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.56
TSHR P16473 2/20 0.53
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
MAPT P10636 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CA2 P00918 3/20 0.47
CA1 P00915 2/20 0.47
CA9 Q16790 1/20 0.47
PLA2G10 O15496 1/20 0.46
PLA2G2A P14555 1/20 0.46
ESR1 P03372 1/20 0.45
ESR2 Q92731 1/20 0.45
PARP1 P09874 1/20 0.44
CYP19A1 P11511 1/20 0.44
FNTA P49354 1/20 0.43
FNTB P49356 1/20 0.43
LIG1 P18858 1/20 0.42
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1004028 0.87 TSHR (0.58) TSHRKDM4EALDH1A1MAPTHPGD
SCHEMBL19439093 0.86 TSHR (0.53) KEAP1TSHRKDM4EALDH1A1MAPT
Hydrochloric Acid SCHEMBL15690391 0.85 TSHR (0.56) TSHRKDM4EALDH1A1MAPTHPGD
SCHEMBL30100451 0.84 TSHR (0.51) TSHRKDM4EALDH1A1MAPTHPGD
SCHEMBL3461077 0.84 TSHR (0.51) TSHRKDM4EALDH1A1MAPTHPGD
SCHEMBL1500536 0.84 TSHR (0.51) TSHRKDM4EALDH1A1MAPTHPGD
SCHEMBL5723969 0.84 CYP19A1 (0.50) TSHRKDM4EALDH1A1MAPTHPGD
SCHEMBL2292722 0.84 TSHR (0.74) KEAP1TSHRALDH1A1CA2CA1
Hydrochloric Acid SCHEMBL29693052 0.83 TSHR (0.50) TSHRKDM4EALDH1A1MAPTHPGD
SCHEMBL7134588 0.82 TSHR (0.54) KEAP1TSHRKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633715-A1 2-(6-AMINO-PYRIDIN-3-YL)-2-HYDROXYETHYLAMINE DERIVATIVES AS BETA 2-ADRENOCEPTORS AGONISTS Pfizer Limited (GB) 2006-03-15 EP disclosed
WO-2004108676-A1 2-(6-AMINO-PYRIDIN-3-YL)-2-HYDROXYETHYLAMINE DERIVATIVES AS BETA 2-ADRENOCEPTORS AGONISTS PFIZER LIMITED (GB) 2004-12-16 WO disclosed