SCHEMBL5728639

SCHEMBL5728639

O=CC(c1ccc(CBr)cc1)C1CCCC1

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.32
PTGS1 P23219 7/20 0.31
PTGS2 P35354 6/20 0.31
MT-CO1 P00395 1/20 0.31
MT-CO2 P00403 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2439182 0.83 NPC1 (0.40) EPHX1
SCHEMBL21368757 0.77 NPC1 (0.41) EPHX1
SCHEMBL6987430 0.77 EPHX1 (0.37) EPHX1
SCHEMBL1515769 0.77 IDO1 (0.46) EPHX1
SCHEMBL6192446 0.76 EPHX1 (0.38) EPHX1
SCHEMBL2442101 0.76 RAB9A (0.44) EPHX1
SCHEMBL6510867 0.76 RAB9A (0.44) EPHX1
SCHEMBL6985435 0.76 EPHX1 (0.39) EPHX1
SCHEMBL193457 0.75 IDO1 (0.49) EPHX1
SCHEMBL8386053 0.74 NPC1 (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed