SCHEMBL5728977

SCHEMBL5728977

CC(C)(C)OC(=O)N1CC2CC1CC2O

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
NR1H2 P55055 1/20 0.43
GPR119 Q8TDV5 4/20 0.41
HSD11B1 P28845 1/20 0.40
PREP P48147 3/20 0.40
CYP1A2 P05177 1/20 0.36
POLB P06746 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
CCR2 P41597 1/20 0.35
F13A1 P00488 1/20 0.35
TGM2 P21980 1/20 0.35
TGM1 P22735 1/20 0.35
AR P10275 1/20 0.34
USP2 O75604 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26906132 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119
SCHEMBL30001283 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119
SCHEMBL29770796 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119
SCHEMBL29827202 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119
SCHEMBL5742486 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119
SCHEMBL29827014 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119
SCHEMBL12276853 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119
SCHEMBL5728974 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119
SCHEMBL20633608 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119
SCHEMBL12274909 1.00 CHRM2 (0.46) CHRM2CHRM1CHRM3NR1H2GPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517708-A1 COMBINATION TREATMENT FOR DEPRESSION AND ANXIETY BY NK1 AND NK3 ANTAGONISTS Pfizer Products Inc. (US) 2005-03-30 EP claimed
WO-2004000355-A1 COMBINATION TREATMENT FOR DEPRESSION AND ANXIETY BY NK1 AND NK3 ANTAGONISTS PFIZER PRODUCTS INC. (US) 2003-12-31 WO claimed
EP-4288426-B1 QUINOXALINE DERIVATIVES AND USES THEREOF BLACK DIAMOND THERAPEUTICS INC (US) 2026-02-04 EP disclosed
EP-4665733-A1 AMINO-SUBSTITUTED PYRROLOTRIAZINE DERIVATIVES AS INHIBITORS OF SGK1 Bristol-Myers Squibb Company (US) 2025-12-24 EP disclosed
US-12447153-B2 HER2 mutation inhibitors PFIZER INC. (US) 2025-10-21 US disclosed
US-20250127907-A1 PARP INHIBITORS Stablix, Inc. 2025-04-24 US disclosed
WO-2025054368-A1 COMPOUNDS, COMPOSITIONS, AND METHODS NICO THERAPEUTICS, INC. (US) 2025-03-13 WO disclosed
CN-115135642-B Inhibitors of EGFR mutant forms 缆图药品公司 2025-03-04 CN disclosed
CN-119431366-A IRAK4 degradation agent compound and application thereof 江苏先声药业有限公司 2025-02-14 CN disclosed
US-20250026736-A1 3-(5-oxy)-1-oxoisoindolin-2-yl)piperidine-2,6-dione Derivatives and Uses thereof NOVARTIS AG (CH) 2025-01-23 US disclosed
WO-2024264072-A2 PARP INHIBITORS Stablix, Inc. (US) 2024-12-26 WO disclosed
EP-0937069-B1 PIPERAZINO DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORP (US) 2006-05-03 EP disclosed
EP-0900204-A4 HETEROCYCLIC COMPOUNDS LILLY CO ELI (US) 2001-03-21 EP disclosed
US-6124312-A ACTIVE DRUG FOR TREATING ALZHEIMER'S DISEASE ELI LILLY AND COMPANY (US) 2000-09-26 US disclosed
US-6051575-A RESPIRATORY SYSTEM DISORDERS; SKIN DISORDERS; ANTIINFLAMMATORY AGENTS SCHERING CORPORATION (US) 2000-04-18 US disclosed
US-5968929-A USEFUL IN THE TREATMENT OF CHRONIC AIRWAY DISEASES SUCH AS ASTHMA SCHERING CORPORATION (US) 1999-10-19 US disclosed
EP-0937069-A1 PIPERAZINO DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1999-08-25 EP disclosed
EP-0900204-A1 HETEROCYCLIC COMPOUNDS ELI LILLY AND COMPANY (US) 1999-03-10 EP disclosed
WO-1998018788-A1 PIPERAZINO DERIVATIVES AS NEUROKININ ANTAGONISTS SCHERING CORPORATION (US) 1998-05-07 WO disclosed
WO-1997040016-A1 HETEROCYCLIC COMPOUNDS ELI LILLY AND COMPANY (US) 1997-10-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250026736-A1 3-(5-oxy)-1-oxoisoindolin-2-yl)piperidine-2,6-dione Derivatives and Uses thereof HBZ, HBG1, HBG2 CHRM2 4722/4885CHRM1 4635/4885CHRM3 4631/4885
US-12447153-B2 HER2 mutation inhibitors ERBB2, EGFR, ERBB3 CHRM2 2009/4885CHRM1 1931/4885CHRM3 3801/4885
US-20250127907-A1 PARP INHIBITORS PARP1, PARP2, PARP3 CHRM2 4885/4885CHRM1 4884/4885CHRM3 4876/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.