SCHEMBL5729327

SCHEMBL5729327

c1cncc(CCCn2cc3ccccc3c2)c1

nearest known ligand 0.55

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.53
TDP1 Q9NUW8 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
HRH1 P35367 2/20 0.50
CHRNA7 P36544 1/20 0.47
TBXAS1 P24557 5/20 0.46
HRH4 Q9H3N8 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
GPR84 Q9NQS5 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29671568 0.81 CYP2A6 (0.58) CYP2A6TDP1L3MBTL1HRH1CHRNA7
SCHEMBL5728469 0.81 HRH1 (0.43) TDP1L3MBTL1HRH1HRH3CYP1A2
SCHEMBL11012977 0.77 CYP11B1 (0.66) CYP2A6TDP1L3MBTL1HRH1TBXAS1
SCHEMBL724788 0.76 TDP1 (0.80) CYP2A6TDP1L3MBTL1HRH1CHRNA7
SCHEMBL29485677 0.76 CYP2A6 (0.76) CYP2A6TDP1L3MBTL1HRH1CHRNA7
SCHEMBL2843094 0.76 CYP2A6 (0.76) CYP2A6TDP1L3MBTL1HRH1CHRNA7
SCHEMBL29485675 0.76 TDP1 (0.80) CYP2A6TDP1L3MBTL1HRH1CHRNA7
SCHEMBL8199794 0.75 TDP1 (0.71) CYP2A6TDP1L3MBTL1HRH1CHRNA7
SCHEMBL8200325 0.75 CYP2A6 (0.68) CYP2A6TDP1L3MBTL1HRH1CHRNA7
SCHEMBL8658187 0.74 HRH1 (0.81) CYP2A6TDP1L3MBTL1HRH1CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644320-A1 INDANE DERIVATES AS MUSCARINIC RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-04-12 EP disclosed
WO-2005009941-A1 INDANE DERIVATES AS MUSCARINIC RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-02-03 WO disclosed