Succinic Acid

Succinic Acid

SCHEMBL5729591

C1=CNc2ccccc2C=C1.O=C(O)CCC(=O)O

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRB1CDK4CDK6CHRM2CHRM3DPP4DRD2DRD3DRD4EGFRHRH1HTR1BHTR1DHTR1FHTR2AHTR2CHTR4SLC6A2SLC6A4

The experimentally established mechanism targets of Succinic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR known ✓ P00533 2/20 0.35
NR4A2 P43354 1/20 0.43
GAA P10253 2/20 0.40
ALDH1A1 P00352 2/20 0.40
CYP2C19 P33261 1/20 0.40
RAB9A P51151 2/20 0.39
FFAR1 O14842 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
HIF1A Q16665 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
KEAP1 Q14145 1/20 0.36
HDAC3 O15379 2/20 0.36
HDAC4 P56524 2/20 0.36
HDAC1 Q13547 2/20 0.36
HDAC7 Q8WUI4 2/20 0.36
HDAC2 Q92769 2/20 0.36
HDAC10 Q969S8 2/20 0.36
HDAC11 Q96DB2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL8507926 0.88 MAPT (0.39) GAAALDH1A1CYP2C19RAB9ASMN1; SMN2
Carbamic Acid SCHEMBL28658378 0.86 MAPT (0.38) GAAALDH1A1CYP2C19RAB9ASMN1; SMN2
SCHEMBL34259 0.84 GAA (0.48) GAAMAPT
Fumaric Acid SCHEMBL4504232 0.83 ALDH1A1 (0.37) GAAALDH1A1CYP2C19RAB9ALMNA
Maleic Acid SCHEMBL4504225 0.83 ALDH1A1 (0.37) GAAALDH1A1CYP2C19RAB9ALMNA
Citric Acid SCHEMBL164689 0.82 ALDH1A1 (0.42) ALDH1A1CYP2C19SMN1; SMN2LMNACYP1A2
Cadaverine Tartrate SCHEMBL3996512 0.82 GAA (0.34) GAARAB9ALMNAMAPTNPC1
Cadaverine Tartrate SCHEMBL3996515 0.82 GAA (0.34) GAARAB9ALMNAMAPTNPC1
Tartaric Acid SCHEMBL30548416 0.82 GAA (0.34) GAARAB9ALMNAMAPTNPC1
Trifluoroacetic Acid SCHEMBL5465747 0.82 CES1 (0.39) GAARAB9AMAPTNPC1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed