SCHEMBL5730007

SCHEMBL5730007

C=Cc1ccc(S(=O)(=O)N2CCN(NC3CCN(c4ccncc4)CC3)C(=O)C2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LSS P48449 2/20 0.43
CYP3A4 P08684 4/20 0.40
CYP2C9 P11712 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C19 P33261 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
HIF1A Q16665 1/20 0.40
CYP17A1 P05093 4/20 0.39
CYP21A2 P08686 4/20 0.39
CYP11B1 P15538 4/20 0.39
F10 P00742 1/20 0.38
MAPK1 P28482 1/20 0.38
F13A1 P00488 1/20 0.37
TGM2 P21980 1/20 0.37
TGM1 P22735 1/20 0.37
CHRM1 P11229 2/20 0.37
CYP19A1 P11511 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5730605 0.87 LSS (0.58) LSSCYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL6797988 0.87 TP53 (0.48) LSSCYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL6891060 0.82 LSS (0.43) LSSCYP3A4CYP2C9CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL6893656 0.82 LSS (0.43) LSSCYP3A4CYP2C9CYP1A2CYP2D6
SCHEMBL5729098 0.80 F10 (0.61) F10
SCHEMBL5729012 0.80 F10 (0.48) LSSF10CHRM1
SCHEMBL5730071 0.80 LSS (0.41) LSSCYP3A4CYP2C9CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL5728956 0.79 F10 (0.47) LSSF10CHRM1
Hydrochloric Acid SCHEMBL5729796 0.79 F10 (0.61) F10
SCHEMBL5730224 0.78 LSS (0.41) LSSSMN1; SMN2MAPK1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1188755-B1 ACYLHYDRAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2006-05-03 EP disclosed
US-6723722-B1 BLOOD COAGULATION FACTOR X INHIBITORS; ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2004-04-20 US disclosed
EP-1188755-A1 ACYLHYDRAZINE DERIVATIVES, PROCESS FOR PREPARING THE SAME AND USE THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-20 EP disclosed