SCHEMBL5730815

SCHEMBL5730815

COCC1CC2N[C@H](CC(c3ccc(CCCOc4c(F)ccc(F)c4Cl)cc3)=C2C(=O)N(Cc2cccc(OC)c2C)C2CC2)C1

nearest known ligand 0.83

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
REN P00797 20/20 0.83
CYP3A4 P08684 2/20 0.81
CTSD P07339 1/20 0.65
CTSE P14091 1/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5925901 1.00 REN (0.83) RENCYP3A4CTSDCTSE
SCHEMBL5730812 1.00 REN (0.83) RENCYP3A4CTSDCTSE
SCHEMBL5729490 0.95 REN (0.80) RENCYP3A4CTSDCTSE
SCHEMBL5925910 0.95 REN (0.80) RENCYP3A4CTSDCTSE
SCHEMBL5729493 0.95 REN (0.80) RENCYP3A4CTSDCTSE
SCHEMBL5925895 0.95 REN (0.83) RENCYP3A4CTSDCTSE
SCHEMBL5729859 0.95 REN (0.83) RENCYP3A4CTSDCTSE
SCHEMBL5729858 0.95 REN (0.83) RENCYP3A4CTSDCTSE
SCHEMBL5925912 0.94 REN (0.83) RENCYP3A4CTSDCTSE
SCHEMBL5823417 0.94 REN (0.83) RENCYP3A4CTSDCTSE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1622907-A1 AZABICYCLONONENE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2006-02-08 EP claimed
WO-2004096803-A1 AZABICYCLONONENE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2004-11-11 WO claimed
EP-1622907-A1 AZABICYCLONONENE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2006-02-08 EP disclosed
WO-2004096803-A1 AZABICYCLONONENE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2004-11-11 WO disclosed