SCHEMBL5731330

SCHEMBL5731330

c1ccc(CNC2=NC(c3ccccc3)CN2c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ATM Q13315 1/20 0.44
ADRA2B P18089 3/20 0.43
ADRA2A P08913 2/20 0.43
ADRA2C P18825 2/20 0.43
NPC1 O15118 1/20 0.40
ALDH1A1 P00352 2/20 0.38
LMNA P02545 2/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CASP3 P42574 2/20 0.38
HRH4 Q9H3N8 1/20 0.36
KDM1A O60341 1/20 0.36
MAOA P21397 1/20 0.36
ALPL P05186 2/20 0.35
ALPI P09923 1/20 0.35
DRD1 P21728 1/20 0.35
KCNH2 Q12809 1/20 0.35
CYP1A2 P05177 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3297432 0.91 MEN1 (0.43) MEN1KMT2AATMADRA2BADRA2A
SCHEMBL3251169 0.91 MEN1 (0.43) MEN1KMT2AATMADRA2BADRA2A
SCHEMBL3255880 0.88 KDM1A (0.45) MEN1KMT2AATMKDM1AMAOA
SCHEMBL3248354 0.88 KDM1A (0.45) MEN1KMT2AATMKDM1AMAOA
SCHEMBL3259028 0.85 ALDH1A1 (0.39) MEN1KMT2AATMALDH1A1HRH4
SCHEMBL3256675 0.85 ALDH1A1 (0.39) MEN1KMT2AATMALDH1A1HRH4
SCHEMBL3254185 0.85 KDM1A (0.48) MEN1KMT2AATMALDH1A1HTT
SCHEMBL3253949 0.85 KDM1A (0.48) MEN1KMT2AATMALDH1A1HTT
SCHEMBL3256393 0.83 KDM1A (0.45) MEN1KMT2AATMNPC1ALDH1A1
SCHEMBL3251081 0.83 KDM1A (0.45) MEN1KMT2AATMNPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006528178-A 2006-12-14 JP claimed
EP-1651613-A1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS Aventis Pharmaceuticals, Inc. (US) 2006-05-03 EP claimed
WO-2005014555-A1 4,5-DIHYDRO-IMIDAZOLE AS P2X7 ION CHANNEL BLOCKERS AVENTIS PHARMACEUTICALS INC. (US) 2005-02-17 WO claimed