SCHEMBL5731390

SCHEMBL5731390

COC1=C(OC)C(=O)C(Cc2cccc(C(=O)N3CCSCC3)c2)=C(C)C1=O

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
NPC1 O15118 2/20 0.45
TP53 P04637 2/20 0.45
RAB9A P51151 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
HPGD P15428 1/20 0.42
PKM P14618 1/20 0.42
PARP1 P09874 9/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
RECQL P46063 1/20 0.40
PDE3B Q13370 1/20 0.40
PDE3A Q14432 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5731705 0.89 NPC1 (0.55) ALDH1A1NPC1TP53RAB9ASMN1; SMN2
SCHEMBL5731269 0.88 HPGD (0.51) ALDH1A1SMN1; SMN2HPGDPKMMEN1
SCHEMBL5732788 0.87 L3MBTL1 (0.56) ALDH1A1NPC1TP53RAB9ASMN1; SMN2
SCHEMBL5730762 0.85 POLB (0.44) ALDH1A1NPC1SMN1; SMN2HTTPKM
SCHEMBL5731389 0.83 L3MBTL1 (0.41) ALDH1A1NPC1SMN1; SMN2LMNAHTT
SCHEMBL5731294 0.82 AR (0.39) ALDH1A1NPC1TP53RAB9ALMNA
SCHEMBL5731108 0.81 TRPV1 (0.51) ALDH1A1SMN1; SMN2LMNAHPGDMEN1
SCHEMBL5731113 0.81 TRPV1 (0.51) ALDH1A1SMN1; SMN2LMNAHPGDMEN1
SCHEMBL5730598 0.79 SMN1; SMN2 (0.47) ALDH1A1SMN1; SMN2LMNAHPGDPKM
SCHEMBL5731206 0.79 MRGPRX4 (0.49) TP53RAB9ASMN1; SMN2PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1008346-B1 NF-kB INHIBITORS CONTAINING BENZOQUINONE DERIVATIVES DAIICHI ASUBIO PHARMA CO LTD (JP) 2006-02-15 EP claimed
US-6703421-B1 ADMINISTERING NF-KAPPA B INHIBITOR DAIICHI SUNTORY PHARMA CO., LTD. (JP) 2004-03-09 US disclosed
EP-1132093-A1 PREVENTIVES OR REMEDIES FOR MYOCARDITIS, DILATED CARDIOMYOPATHY AND CARDIAC INSUFFICIENCY CONTAINING NF-KAPPA B INHIBITORS AS THE ACTIVE INGREDIENT SUNTORY LIMITED (JP) 2001-09-12 EP disclosed