SCHEMBL5731471

SCHEMBL5731471

CCCCn1c(O)nc2c(N)ncnc21

nearest known ligand 0.70

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 7/20 0.70
ADORA2B P29275 6/20 0.70
ADORA1 P30542 6/20 0.70
HSP90B1 P14625 1/20 0.56
ADORA3 P0DMS8 3/20 0.55
HSP90AA1 P07900 7/20 0.53
HSP90AB1 P08238 7/20 0.53
ERBB2 P04626 6/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20878863 0.84 ADORA2A (0.72) ADORA2AADORA2BADORA1HSP90B1ADORA3
SCHEMBL1965296 0.82 ADORA2A (1.00) ADORA2AADORA2BADORA1HSP90B1ADORA3
SCHEMBL29157955 0.78 ADORA2A (0.64) ADORA2AADORA2BADORA1HSP90B1ADORA3
SCHEMBL5072517 0.77 ADORA2A (0.85) ADORA2AADORA2BADORA1HSP90B1ADORA3
SCHEMBL5732048 0.76 ADORA2A (0.72) ADORA2AADORA2BADORA1ADORA3
SCHEMBL2980005 0.76 ADORA2A (0.64) ADORA2AADORA2BADORA1ADORA3
SCHEMBL1966178 0.74 HSP90AA1 (0.75) HSP90B1HSP90AA1HSP90AB1ERBB2
SCHEMBL14044861 0.74 HSP90AA1 (0.83) ADORA2AADORA2BADORA1HSP90AA1HSP90AB1
SCHEMBL22359153 0.74 ADORA2A (0.59) ADORA2AADORA2BADORA1HSP90B1ADORA3
SCHEMBL30503500 0.74 ADORA2A (0.59) ADORA2AADORA2BADORA1HSP90B1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1043021-B1 PURINE DERIVATIVES FOR THE TREATMENT OF ALLERGIC DISEASES AND SYSTEMIC LUPUS ERYTHEMATOSUS DAINIPPON SUMITOMO PHARMA CO (JP) 2006-05-03 EP disclosed
EP-0882727-B9 NOVEL PURINE DERIVATIVES SUMITOMO PHARMA (JP) 2005-06-15 EP disclosed
EP-0882727-B1 NOVEL PURINE DERIVATIVES SUMITOMO PHARMA (JP) 2004-12-01 EP disclosed
US-6376501-B1 INHIBITING OR REGULATING IMMUNE RESPONSE USING PURINE-DERIVED COMPOUND; NON-STEROIDAL COMPOUND JAPAN ENERGY CORPORATION (JP) 2002-04-23 US disclosed
EP-1043021-A1 TYPE 2 HELPER T CELL-SELECTIVE IMMUNE RESPONSE SUPPRESSORS Japan Energy Corporation (JP) 2000-10-11 EP disclosed
US-6028076-A FOR INDUCING .ALPHA.-INTERFERON IN A PATIENT HAVING HEPATITIS B OR C, BY ADMINISTERING PURINE DERIVATIVE JAPAN ENERGY CORPORATION (JP) 2000-02-22 US disclosed
EP-0882727-A1 NOVEL PURINE DERIVATIVES JAPAN ENERGY CORPORATION (JP) 1998-12-09 EP disclosed