SCHEMBL5732504

SCHEMBL5732504

CC(C)(C)OC(=O)NC(CCc1ccccc1)C(=O)NCC(=O)O

nearest known ligand 0.77

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 13/20 0.77
CTSK P43235 13/20 0.77
CTSB P07858 4/20 0.59
CTSL P07711 2/20 0.59
AKT1 P31749 1/20 0.52
SCN9A Q15858 1/20 0.51
PPARA Q07869 2/20 0.49
PPARG P37231 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5732509 1.00 CTSS (0.77) CTSSCTSKCTSBCTSLAKT1
SCHEMBL5564256 0.92 CTSS (0.75) CTSSCTSKCTSBCTSLAKT1
SCHEMBL5564249 0.92 CTSS (0.75) CTSSCTSKCTSBCTSLAKT1
SCHEMBL20814294 0.89 CTSS (0.62) CTSSCTSKCTSBCTSLAKT1
SCHEMBL15989226 0.88 CTSS (0.77) CTSSCTSKCTSBCTSLAKT1
SCHEMBL2793925 0.88 CTSS (0.76) CTSSCTSKCTSBCTSLAKT1
SCHEMBL1001781 0.88 CTSS (0.76) CTSSCTSKCTSBCTSLAKT1
SCHEMBL3758017 0.87 CTSS (0.75) CTSSCTSKCTSBCTSLAKT1
SCHEMBL3763891 0.87 CTSS (0.75) CTSSCTSKCTSBCTSLAKT1
SCHEMBL4374188 0.86 CTSS (0.74) CTSSCTSKCTSBCTSLSCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664063-A1 SUBSTITUTED PIPERAZINES OF AZEPINES, OXAZEPINES, AND THIAZEPINES ELI LILLY AND COMPANY (US) 2006-06-07 EP disclosed
WO-2005026177-A1 SUBSTITUTED PIPERAZINES OF AZEPINES, OXAZEPINES, AND THIAZEPINES ELI LILLY AND COMPANY (US) 2005-03-24 WO disclosed