SCHEMBL5735015

SCHEMBL5735015

CC(C)N(Cc1ccc(C(=O)C2CCNCC2)cc1)C(C)C

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.56
CYP2D6 P10635 1/20 0.56
KMT2A Q03164 1/20 0.56
HDAC1 Q13547 1/20 0.51
HDAC8 Q9BY41 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
SLC6A2 P23975 10/20 0.41
SLC6A4 P31645 10/20 0.41
SLC6A3 Q01959 4/20 0.40
ALDH1A1 P00352 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KHK P50053 1/20 0.38
OPRD1 P41143 1/20 0.38
KCNH2 Q12809 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7036133 0.84 MEN1 (0.60) MEN1CYP2D6KMT2AHDAC6SLC6A2
Hydrochloric Acid SCHEMBL20838548 0.83 MEN1 (0.63) MEN1CYP2D6KMT2AHDAC6SLC6A2
SCHEMBL20883790 0.79 MEN1 (0.66) MEN1CYP2D6KMT2AALDH1A1SMN1; SMN2
SCHEMBL6622933 0.77 MEN1 (0.62) MEN1CYP2D6KMT2AALDH1A1SMN1; SMN2
SCHEMBL4038817 0.76 MEN1 (0.66) MEN1CYP2D6KMT2ASLC6A2SLC6A4
SCHEMBL5733737 0.75 HRH3 (0.54) MEN1KMT2AHDAC1HDAC8HDAC6
Hydrochloric Acid SCHEMBL27829790 0.75 MEN1 (0.64) MEN1CYP2D6KMT2AHDAC6ALDH1A1
SCHEMBL5735422 0.74 MGLL (0.44) MEN1KMT2AHDAC1HDAC8HDAC6
SCHEMBL1582773 0.74 KMT2A (0.96) MEN1CYP2D6KMT2AALDH1A1KHK
SCHEMBL28750644 0.74 MEN1 (0.58) MEN1CYP2D6KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986551-B1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA PHARMACEUTICAL (JP) 2006-08-02 EP disclosed
US-6359134-B1 ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-03-19 US disclosed
EP-0986551-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Pharmaceutical Company Limited (JP) 2000-03-22 EP disclosed
WO-1998054164-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-12-03 WO disclosed