SCHEMBL5735112

SCHEMBL5735112

CCOc1cccc(-c2cc(=O)n(C)c3c(C(N)(c4ccc(Cl)cc4)c4cncn4C)cccc23)c1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
FNTA P49354 13/20 0.52
FNTB P49356 13/20 0.52
PGGT1B P53609 3/20 0.52
CYP3A4 P08684 6/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6174338 0.92 FNTA (0.44) FNTAFNTBPGGT1BCYP3A4
SCHEMBL5737090 0.90 FNTA (0.59) FNTAFNTBPGGT1BCYP3A4
SCHEMBL5071351 0.88 FNTA (0.64) FNTAFNTBPGGT1BCYP3A4
SCHEMBL5734468 0.86 CYP3A4 (0.53) FNTAFNTBPGGT1BCYP3A4
SCHEMBL1683530 0.86 CYP3A4 (0.67) FNTAFNTBPGGT1BCYP3A4
SCHEMBL6172596 0.84 FNTA (0.49) FNTAFNTBPGGT1BCYP3A4
SCHEMBL6173339 0.82 FNTA (0.55) FNTAFNTBPGGT1BCYP3A4
SCHEMBL6171352 0.82 FNTA (0.45) FNTAFNTBPGGT1BCYP3A4
SCHEMBL6172263 0.81 FNTA (0.54) FNTAFNTBPGGT1BCYP3A4
SCHEMBL6170815 0.79 CYP3A4 (0.48) FNTAFNTBPGGT1BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1162201-B1 Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives JANSSEN PHARMACEUTICA NV (BE) 2006-03-29 EP claimed
EP-1094815-B1 FARNESYL PROTEIN TRANSFERASE INHIBITORS FOR TREATING ARTHROPATHIES JANSSEN PHARMACEUTICA NV (BE) 2003-11-12 EP claimed
EP-1094839-B1 FARNESYL PROTEIN TRANSFERASE INHIBITORS WITH (IN VIVO) RADIOSENSITIZING PROPERTIES JANSSEN PHARMACEUTICA NV (BE) 2003-05-02 EP claimed
EP-0865440-B1 FARNESYL PROTEIN TRANSFERASE INHIBITING (IMIDAZOL-5-YL)METHYL-2-QUINOLINONE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2002-04-03 EP claimed