SCHEMBL5736839

SCHEMBL5736839

CCc1nc(-c2ccncc2)sc1C(=O)N1CCN(S(=O)(=O)c2ccc3cc(Cl)ccc3c2)CC1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
F10 P00742 16/20 0.51
ATM Q13315 1/20 0.51
F2 P00734 3/20 0.51
LMNA P02545 1/20 0.45
GAA P10253 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
THRA P10827 1/20 0.45
THRB P10828 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5734576 0.90 SMN1; SMN2 (0.51) F10ATMF2LMNASMN1; SMN2
SCHEMBL5734359 0.89 F10 (0.54) F10ATMF2LMNAGAA
SCHEMBL5737962 0.80 F10 (0.57) F10ATMF2LMNAGAA
SCHEMBL5734441 0.80 F10 (0.56) F10ATMF2LMNAGAA
SCHEMBL5735531 0.80 MAPT (0.53) ATMLMNASMN1; SMN2
SCHEMBL5734474 0.79 ATM (0.66) ATMLMNAGAASMN1; SMN2
SCHEMBL5737352 0.79 SMN1; SMN2 (0.54) F10ATMF2LMNASMN1; SMN2
SCHEMBL5193868 0.79 ATM (0.71) F10ATMF2LMNAGAA
SCHEMBL5735064 0.78 LSS (0.54) LMNAGAASMN1; SMN2THRATHRB
SCHEMBL5734701 0.78 F10 (0.56) F10ATMF2LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986551-B1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA PHARMACEUTICAL (JP) 2006-08-02 EP disclosed
US-6359134-B1 ANTICOAGULANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-03-19 US disclosed
EP-0986551-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE Takeda Pharmaceutical Company Limited (JP) 2000-03-22 EP disclosed
WO-1998054164-A1 SULFONAMIDE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-12-03 WO disclosed