SCHEMBL5736856

SCHEMBL5736856

Cn1cncc1C(O)(c1ccc(Cl)cc1)c1cccc2c(-c3cccc(Cl)c3)cc(=O)n(C)c12

nearest known ligand 0.73

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FNTA P49354 15/20 0.73
FNTB P49356 15/20 0.73
PGGT1B P53609 1/20 0.55
CYP3A4 P08684 2/20 0.50
RORC P51449 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6172284 0.89 FNTA (0.61) FNTAFNTBPGGT1BCYP3A4RORC
SCHEMBL5737090 0.89 FNTA (0.59) FNTAFNTBPGGT1BCYP3A4RORC
SCHEMBL5071351 0.88 FNTA (0.64) FNTAFNTBPGGT1BCYP3A4
SCHEMBL6167630 0.86 FNTA (0.62) FNTAFNTBPGGT1BCYP3A4RORC
SCHEMBL5755627 0.85 FNTA (0.55) FNTAFNTBPGGT1BCYP3A4RORC
SCHEMBL5755701 0.85 FNTA (0.54) FNTAFNTBPGGT1BCYP3A4RORC
SCHEMBL1682772 0.85 FNTA (1.00) FNTAFNTBCYP3A4
SCHEMBL13928075 0.85 FNTA (1.00) FNTAFNTBCYP3A4
SCHEMBL6171125 0.84 FNTA (0.55) FNTAFNTBPGGT1BCYP3A4RORC
Hydrochloric Acid SCHEMBL6435591 0.84 FNTA (0.98) FNTAFNTBCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1162201-B1 Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives JANSSEN PHARMACEUTICA NV (BE) 2006-03-29 EP claimed
EP-1094815-B1 FARNESYL PROTEIN TRANSFERASE INHIBITORS FOR TREATING ARTHROPATHIES JANSSEN PHARMACEUTICA NV (BE) 2003-11-12 EP claimed
EP-1094839-B1 FARNESYL PROTEIN TRANSFERASE INHIBITORS WITH (IN VIVO) RADIOSENSITIZING PROPERTIES JANSSEN PHARMACEUTICA NV (BE) 2003-05-02 EP claimed
EP-0865440-B1 FARNESYL PROTEIN TRANSFERASE INHIBITING (IMIDAZOL-5-YL)METHYL-2-QUINOLINONE DERIVATIVES JANSSEN PHARMACEUTICA NV (BE) 2002-04-03 EP claimed