SCHEMBL5737270

SCHEMBL5737270

COc1ccc(-c2noc(-c3ccc(O)cc3)c2-c2[c]ccc(OCCC3CCCCN3)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.42
SSTR2 P30874 5/20 0.38
CHEK2 O96017 1/20 0.37
PTGS2 P35354 4/20 0.37
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
MERTK Q12866 1/20 0.33
PTGS1 P23219 1/20 0.33
PDE3A Q14432 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HIF1A Q16665 1/20 0.33
PHLPP2 Q6ZVD8 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5729709 0.83 CHEK2 (0.44) CHEK1SSTR2CHEK2PTGS2
SCHEMBL5730047 0.83 CHEK2 (0.44) CHEK1SSTR2CHEK2PTGS2
SCHEMBL6394083 0.83 PTGS2 (0.47) CHEK1CHEK2PTGS2MERTKPTGS1
SCHEMBL5729300 0.83 PTGS2 (0.47) CHEK1CHEK2PTGS2MERTKPTGS1
SCHEMBL7662650 0.79 CHEK2 (0.42) CHEK1SSTR2CHEK2PTGS2AURKB
SCHEMBL5729507 0.79 CHEK2 (0.46) CHEK1SSTR2CHEK2PTGS2
SCHEMBL5729625 0.79 CHEK2 (0.46) CHEK1SSTR2CHEK2PTGS2
SCHEMBL5729577 0.79 CHEK1 (0.42) CHEK1SSTR2CHEK2PTGS2CHRNB4
Hydrochloric Acid SCHEMBL6311273 0.79 CHEK1 (0.42) CHEK1SSTR2CHEK2PTGS2CHRNB4
SCHEMBL5729040 0.75 CHEK2 (0.48) CHEK1SSTR2CHEK2PTGS2MERTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1102755-B1 SUBSTITUTED ISOXAZOLE DERIVATIVES AS ESTROGEN RECEPTOR MODULATORS CHIRON CORP (US) 2006-01-04 EP claimed