SCHEMBL5737489

SCHEMBL5737489

Cc1cccc(NS(=O)(=O)c2ccc(NC(=O)[C@@](C)(O)C(F)(F)F)c(Cl)c2)c1

nearest known ligand 0.66

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGES2 Q9H7Z7 1/20 0.66
PDK1 Q15118 17/20 0.64
PDK2 Q15119 17/20 0.64
PDK3 Q15120 17/20 0.64
PDK4 Q16654 17/20 0.64
NR1H2 P55055 1/20 0.56
NR1H3 Q13133 1/20 0.56
ABCB11 O95342 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5739088 0.91 PTGES2 (0.67) PTGES2PDK1PDK2PDK3PDK4
SCHEMBL5748675 0.89 PTGES2 (0.74) PTGES2PDK1PDK2PDK3PDK4
SCHEMBL5735945 0.89 PTGES2 (0.65) PTGES2PDK1PDK2PDK3PDK4
SCHEMBL5737233 0.89 PTGES2 (0.65) PTGES2PDK1PDK2PDK3PDK4
SCHEMBL5736462 0.89 PTGES2 (0.65) PTGES2PDK1PDK2PDK3PDK4
SCHEMBL5737922 0.89 PDK1 (0.68) PTGES2PDK1PDK2PDK3PDK4
SCHEMBL5737307 0.87 PDK1 (0.65) PTGES2PDK1PDK2PDK3PDK4
SCHEMBL5738183 0.86 PDK1 (0.68) PTGES2PDK1PDK2PDK3PDK4
SCHEMBL6357232 0.86 NR1H2 (0.65) PTGES2PDK1PDK2PDK3PDK4
SCHEMBL5738271 0.85 PDK1 (0.69) PTGES2PDK1PDK2PDK3PDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1064274-B1 BENZENESULFONAMIDE DERIVATIVES AND THEIR USE AS MEDICAMENTS ASTRAZENECA AB (SE) 2006-04-19 EP disclosed