SCHEMBL5740256

SCHEMBL5740256

Cc1c(OC(=O)O)cn2ncnc(C3C(=O)Nc4ccccc43)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.35
ALDH1A1 P00352 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
GAA P10253 1/20 0.34
IDO1 P14902 4/20 0.34
TDO2 P48775 2/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
POLB P06746 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
HPGDS O60760 1/20 0.32
MAP2K1 Q02750 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14451971 0.93 ALDH1A1 (0.35) MAPTALDH1A1L3MBTL1GAAIDO1
SCHEMBL5740055 0.91 MAPT (0.35) MAPTALDH1A1L3MBTL1GAAIDO1
SCHEMBL4047213 0.89 PDE4A (0.41) MAPTALDH1A1L3MBTL1GAAIDO1
SCHEMBL14452013 0.86 POLB (0.41) MAPTL3MBTL1IDO1TDO2POLB
SCHEMBL1462071 0.85 MAPK14 (0.38) MAPTALDH1A1L3MBTL1IDO1TDO2
SCHEMBL1459917 0.83 MAPK14 (0.39) MAPTALDH1A1L3MBTL1GAAIDO1
SCHEMBL4048478 0.83 KDR (0.47) MAP2K1
SCHEMBL4052257 0.83 IDO1 (0.34) MAPTALDH1A1L3MBTL1GAAIDO1
SCHEMBL5740098 0.82 ALDH1A1 (0.41) MAPTALDH1A1L3MBTL1GAAPOLB
SCHEMBL5739045 0.81 ALDH1A1 (0.41) MAPTALDH1A1L3MBTL1GAAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed