Bicarbonate

Bicarbonate

SCHEMBL5740452

O=C(O)O.O=C1COc2ccc(CN[C@H]3C=C[C@@H](O)CC3)nc2N1

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 17/20 0.48
KCNQ1 P51787 1/20 0.41
CACNA1C Q13936 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL5749485 1.00 KCNH2 (0.48) KCNH2KCNQ1CACNA1C
SCHEMBL5740447 0.84 KCNH2 (0.49) KCNH2
SCHEMBL5739490 0.84 KCNH2 (0.49) KCNH2
Bicarbonate SCHEMBL5738348 0.80 KCNH2 (0.40) KCNH2
Bicarbonate SCHEMBL5738279 0.80 KCNH2 (0.40) KCNH2
Bicarbonate SCHEMBL4045503 0.80 KCNH2 (0.47) KCNH2
Bicarbonate SCHEMBL4054052 0.80 KCNH2 (0.47) KCNH2
SCHEMBL17956688 0.79 KCNH2 (0.45) KCNH2
SCHEMBL5262019 0.78 KCNH2 (0.54) KCNH2KCNQ1CACNA1C
SCHEMBL5262012 0.78 KCNH2 (0.54) KCNH2KCNQ1CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539133-B1 AMINOCYCLOHEXENE QUINOLINES AND THEIR AZAISOSTERIC ANALOGUES WITH ANTIBACTERIAL ACTIVITY GLAXO GROUP LTD (GB) 2006-08-23 EP claimed