SCHEMBL5740994

SCHEMBL5740994

Nc1nc(Nc2ccc3nc(-c4cccc(Cl)c4)cc(N)c3c2)cc(C(F)(F)F)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.47
AGPAT2 O15120 3/20 0.47
KDM4E B2RXH2 2/20 0.44
HSD17B10 Q99714 2/20 0.44
ALDH1A1 P00352 1/20 0.42
MCHR1 Q99705 1/20 0.42
ACP1 P24666 4/20 0.41
ROCK2 O75116 1/20 0.41
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
HRH4 Q9H3N8 1/20 0.39
MAP4K4 O95819 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
PDE4B Q07343 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5742129 0.90 KDM4E (0.55) AGPAT2KDM4EHSD17B10ALDH1A1MCHR1
SCHEMBL5740513 0.89 KDM4E (0.44) AGPAT2KDM4EHSD17B10MCHR1ROCK2
SCHEMBL5744288 0.89 KDM4E (0.56) AGPAT2KDM4EHSD17B10ALDH1A1MCHR1
SCHEMBL5742792 0.89 AGPAT2 (0.59) AGPAT2ACP1TP53MAPTHRH4
SCHEMBL5741884 0.88 AGPAT2 (0.52) AGPAT2MCHR1ACP1ROCK2LMNA
SCHEMBL5741026 0.88 AGPAT2 (0.52) AGPAT2MCHR1ACP1ROCK2LMNA
SCHEMBL5742859 0.87 AGPAT2 (0.63) AGPAT2KDM4EACP1TP53MAPT
SCHEMBL5743344 0.85 AGPAT2 (0.53) AGPAT2ACP1ROCK2MAPTHRH4
SCHEMBL5741974 0.85 AGPAT2 (0.53) AGPAT2ACP1ROCK2MAPTHRH4
SCHEMBL5742786 0.85 AGPAT2 (0.64) AGPAT2ACP1TP53MAPTHRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed