SCHEMBL5744288

SCHEMBL5744288

Nc1nc(Nc2ccc3nc(-c4ccc(Cl)cc4)cc(N)c3c2)cc(C(F)(F)F)n1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.56
HSD17B10 Q99714 2/20 0.56
ALDH1A1 P00352 1/20 0.56
AGPAT2 O15120 6/20 0.52
NPC1 O15118 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
RAB9A P51151 1/20 0.42
MCHR1 Q99705 2/20 0.41
ACHE P22303 1/20 0.41
ROCK2 O75116 1/20 0.40
DOT1L Q8TEK3 1/20 0.40
TERT O14746 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
PTGS2 P35354 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5743755 0.91 KDM4E (0.55) KDM4EHSD17B10ALDH1A1AGPAT2MCHR1
SCHEMBL5742129 0.90 KDM4E (0.55) KDM4EHSD17B10ALDH1A1AGPAT2MCHR1
SCHEMBL5740994 0.89 PDE4D (0.47) KDM4EHSD17B10ALDH1A1AGPAT2CYP3A4
SCHEMBL5741991 0.89 AGPAT2 (0.57) KDM4EHSD17B10ALDH1A1AGPAT2NPC1
SCHEMBL5742875 0.89 AGPAT2 (0.57) KDM4EHSD17B10ALDH1A1AGPAT2NPC1
SCHEMBL5742668 0.87 KDM4E (0.58) KDM4EHSD17B10ALDH1A1RAB9AACHE
SCHEMBL5740139 0.85 AGPAT2 (0.60) KDM4EHSD17B10ALDH1A1AGPAT2NPC1
SCHEMBL5741862 0.84 AGPAT2 (0.57) KDM4EHSD17B10ALDH1A1AGPAT2MCHR1
SCHEMBL5740513 0.84 KDM4E (0.44) KDM4EHSD17B10AGPAT2MCHR1ACHE
SCHEMBL5740529 0.83 MCHR1 (0.53) AGPAT2MCHR1ROCK2DOT1LTERT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339706-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-04-19 EP disclosed