SCHEMBL5741016

SCHEMBL5741016

CCOC(=O)Oc1cn2ncnc(C3C(=O)Nc4ccccc43)c2c1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 5/20 0.40
ALDH1A1 P00352 4/20 0.40
MAPT P10636 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 3/20 0.38
HTT P42858 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
USP2 O75604 1/20 0.37
MAPK1 P28482 1/20 0.37
KDM4E B2RXH2 2/20 0.35
TSHR P16473 3/20 0.35
EGFR P00533 1/20 0.35
ERBB2 P04626 1/20 0.35
PKM P14618 1/20 0.34
MAP2K1 Q02750 1/20 0.34
GSK3A P49840 1/20 0.33
GSK3B P49841 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740098 0.95 ALDH1A1 (0.41) HSD17B10ALDH1A1MAPTL3MBTL1GAA
SCHEMBL5739045 0.94 ALDH1A1 (0.41) HSD17B10ALDH1A1MAPTL3MBTL1GAA
SCHEMBL5738339 0.88 ALDH1A1 (0.41) HSD17B10ALDH1A1MAPTL3MBTL1GAA
SCHEMBL4044556 0.87 PDE4A (0.41) HSD17B10ALDH1A1MAPTL3MBTL1GAA
SCHEMBL14470113 0.86 ALDH1A1 (0.40) HSD17B10ALDH1A1MAPTL3MBTL1GAA
SCHEMBL4049523 0.84 HSD17B10 (0.40) HSD17B10ALDH1A1MAPTTSHRPDE4A
SCHEMBL4044212 0.84 KDR (0.47) ALDH1A1MAPTL3MBTL1MEN1KMT2A
SCHEMBL5740055 0.83 MAPT (0.35) HSD17B10ALDH1A1MAPTL3MBTL1GAA
SCHEMBL4044576 0.83 PDE4A (0.39) HSD17B10ALDH1A1MAPTL3MBTL1GAA
SCHEMBL4041795 0.81 PDE4A (0.34) HSD17B10ALDH1A1MAPTL3MBTL1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed