SCHEMBL5741316

SCHEMBL5741316

CC(C)Cc1cccc(O)c1C(=N)N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.53
GABRB2 P47870 2/20 0.53
ELANE P08246 1/20 0.39
CTSG P08311 1/20 0.39
CA12 O43570 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA7 P43166 2/20 0.37
CA9 Q16790 2/20 0.37
CA14 Q9ULX7 2/20 0.37
THRB P10828 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
TAS1R2 Q8TE23 1/20 0.34
BID P55957 3/20 0.33
MCL1 Q07820 3/20 0.33
BCL2L1 Q07817 2/20 0.33
BAK1 Q16611 2/20 0.33
POLB P06746 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5743029 0.83 GABRA1 (0.53) GABRA1GABRB2ELANECTSGCA12
SCHEMBL5744962 0.81 BID (0.42) GABRA1GABRB2BIDMCL1BCL2L1
SCHEMBL20806632 0.78 GABRA1 (0.43) GABRA1GABRB2GRIN2DGRIN3BGRIN1
SCHEMBL4963083 0.77 BID (0.55) GABRA1GABRB2CA12CA1CA2
SCHEMBL5742072 0.77 BID (0.47) ELANECTSGCA12CA1CA2
SCHEMBL6675604 0.74 GABRA1 (0.61) GABRA1GABRB2ELANECTSGPOLB
SCHEMBL1053654 0.74 GABRA1 (0.79) GABRA1GABRB2ELANECTSGCA1
SCHEMBL11393106 0.73 BID (0.63) BIDMCL1BCL2L1BAK1
SCHEMBL108067 0.73 GABRA1 (0.64) GABRA1GABRB2ELANECTSGCA12
SCHEMBL258656 0.72 GABRA1 (0.63) GABRA1GABRB2ELANECTSGPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678146-A1 PYRIMIDINE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION Pharmacia Corporation (US) 2006-07-12 EP disclosed
WO-2005040133-A1 PYRIMIDINE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA CORPORATION (US) 2005-05-06 WO disclosed