SCHEMBL5741504

SCHEMBL5741504

C=CC1C[C@@]1(NC(=O)[C@@H]1C[C@@H](Oc2cc(-c3ccccc3)nc3cc(OC)ccc23)CN1C(=O)NN)C(=O)OCC

nearest known ligand 0.45

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSB P07858 2/20 0.39
PPP3CB P16298 1/20 0.39
CYP3A4 P08684 1/20 0.39
ADAM17 P78536 2/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TACR3 P29371 6/20 0.36
TDP1 Q9NUW8 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3041937 1.00 CTSB (0.39) CTSBPPP3CBCYP3A4ADAM17KDM4E
SCHEMBL3041949 1.00 CTSB (0.39) CTSBPPP3CBCYP3A4ADAM17KDM4E
SCHEMBL5741505 1.00 CTSB (0.39) CTSBPPP3CBCYP3A4ADAM17KDM4E
SCHEMBL13519865 1.00 CTSB (0.39) CTSBPPP3CBCYP3A4ADAM17KDM4E
SCHEMBL3042218 0.94 CTSB (0.39) CTSBPPP3CBCYP3A4ADAM17KDM4E
SCHEMBL4979076 0.94 CTSB (0.41) CTSBPPP3CBCYP3A4ADAM17KDM4E
SCHEMBL14282972 0.93 CTSB (0.40) CTSBPPP3CBCYP3A4ADAM17KDM4E
SCHEMBL14282971 0.93 CTSB (0.40) CTSBPPP3CBCYP3A4ADAM17KDM4E
SCHEMBL13672819 0.92 CTSB (0.43) CTSBPPP3CBCYP3A4KDM4EALDH1A1
SCHEMBL3053155 0.92 CTSB (0.43) CTSBPPP3CBCYP3A4KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713822-A2 HCV NS-3 SERINE PROTEASE INHIBITORS Medivir Aktiebolag (SE) 2006-10-25 EP disclosed
WO-2005073216-A2 HCV NS-3 SERINE PROTEASE INHIBITORS MEDIVIR AB (SE) 2005-08-11 WO disclosed