SCHEMBL5742985

SCHEMBL5742985

NC(=O)Nc1ccc(C(F)(F)F)c(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.57
PDK1 Q15118 1/20 0.51
KIF11 P52732 4/20 0.50
NPC1 O15118 2/20 0.50
HSD11B1 P28845 1/20 0.48
CA1 P00915 3/20 0.48
CA2 P00918 3/20 0.48
CA7 P43166 3/20 0.48
CA9 Q16790 3/20 0.48
SMN1; SMN2 Q16637 2/20 0.47
MEN1 O00255 1/20 0.47
LMNA P02545 1/20 0.47
HSP90AA1 P07900 1/20 0.47
MAPT P10636 1/20 0.47
NPY1R P25929 1/20 0.47
HTT P42858 1/20 0.47
NPY2R P49146 1/20 0.47
RAB9A P51151 1/20 0.47
KMT2A Q03164 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2457115 0.87 KDR (0.76) KDRPDK1CA1CA2CA7
SCHEMBL29759440 0.87 KDR (0.76) KDRPDK1CA1CA2CA7
SCHEMBL11245874 0.86 KDR (0.50) KDRPDK1NPC1CA1CA2
SCHEMBL4556067 0.86 KDR (0.75) KDRPDK1NPC1CA1CA2
SCHEMBL5248618 0.85 KDR (0.58) KDRPDK1CA1CA2CA7
SCHEMBL11787916 0.85 KDR (0.58) KDRPDK1CA1CA2CA7
Fluoride SCHEMBL11787921 0.83 KDR (0.57) KDRPDK1CA1CA2CA7
SCHEMBL28875490 0.83 KDR (0.57) KDRPDK1KIF11SMN1; SMN2MEN1
SCHEMBL23194458 0.82 KDR (0.55) KDRPDK1SMN1; SMN2NPSR1FLT1
SCHEMBL1943274 0.82 KDR (0.55) KDRPDK1CA1CA2CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1727541-A1 IMIDAZOLE-BASED HMG-COA REDUCTASE INHIBITORS Warner-Lambert Company LLC (US) 2006-12-06 EP disclosed
WO-2006059210-A2 FUSED BICYCLIC PYRROLS AS HMG-COA REDUCTASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2006-06-08 WO disclosed
WO-2005079790-A1 IMIDAZOLE-BASED HMG-COA REDUCTASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2005-09-01 WO disclosed