SCHEMBL11245874

SCHEMBL11245874

N=C(NC(N)=O)Nc1ccc(C(F)(F)F)c(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.50
PDK1 Q15118 1/20 0.49
FLT1 P17948 6/20 0.45
TMPRSS4 Q9NRS4 2/20 0.44
GRM4 Q14833 1/20 0.44
MEN1 O00255 2/20 0.43
HTT P42858 2/20 0.43
KMT2A Q03164 2/20 0.43
NPSR1 Q6W5P4 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA7 P43166 2/20 0.43
CA9 Q16790 2/20 0.43
TRPV1 Q8NER1 2/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
HSP90AA1 P07900 1/20 0.42
MAPT P10636 1/20 0.42
NPY1R P25929 1/20 0.42
NPY2R P49146 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5742985 0.86 KDR (0.57) KDRPDK1FLT1TMPRSS4GRM4
SCHEMBL11259118 0.84 KCNQ3 (0.45) KDRPDK1TMPRSS4GRM4HTT
SCHEMBL4100753 0.83 EPHX1 (0.58) GRM4MEN1HTTKMT2ANPSR1
SCHEMBL11254366 0.83 MAPT (0.47) KDRPDK1TMPRSS4MEN1HTT
SCHEMBL4103669 0.82 SLC2A1 (0.56) MEN1HTTKMT2ANPSR1CA2
SCHEMBL11263943 0.82 HTT (0.46) KDRPDK1FLT1TMPRSS4MEN1
SCHEMBL11257942 0.81 HTT (0.58) KDRPDK1MEN1HTTKMT2A
SCHEMBL4556067 0.80 KDR (0.75) KDRPDK1MEN1HTTKMT2A
SCHEMBL6699635 0.79 MAOB (0.47) MEN1KMT2ANPC1MAPTRAB9A
SCHEMBL11253702 0.79 PLAU (0.46) MEN1KMT2ANPSR1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4326074-A ANTIDIARRHEA AGENTS WILLIAM H. RORER, INC. (US) 1982-04-20 US disclosed
US-4115564-A Treatment of diarrhea with amidinoureas WILLIAM H. RORER, INC. (US) 1978-09-19 US disclosed