SCHEMBL574340

SCHEMBL574340

C=CCOc1cccc2cccnc12

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.55
RAB9A P51151 5/20 0.55
LMNA P02545 5/20 0.54
NPC1 O15118 4/20 0.54
MEN1 O00255 4/20 0.54
KMT2A Q03164 4/20 0.54
SMN1; SMN2 Q16637 3/20 0.54
GAA P10253 2/20 0.53
MAPK1 P28482 2/20 0.53
KDM4E B2RXH2 5/20 0.51
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
POLB P06746 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9051415 0.83 MAPT (0.60) MAPTRAB9ALMNANPC1MEN1
SCHEMBL5215459 0.83 RAB9A (0.55) MAPTRAB9ALMNANPC1MEN1
SCHEMBL5586004 0.80 RAB9A (0.60) MAPTRAB9ALMNANPC1MEN1
SCHEMBL10367557 0.80 MAPT (0.53) MAPTRAB9ALMNANPC1MEN1
SCHEMBL10367558 0.80 MAPT (0.53) MAPTRAB9ALMNANPC1MEN1
SCHEMBL8027680 0.79 MAPT (0.54) MAPTRAB9ALMNANPC1MEN1
SCHEMBL8027893 0.79 SMN1; SMN2 (0.54) MAPTRAB9ALMNANPC1MEN1
SCHEMBL10365652 0.79 MEN1 (0.57) MAPTLMNAMEN1KMT2ASMN1; SMN2
SCHEMBL7869387 0.79 KDM4E (0.53) MAPTRAB9ALMNANPC1MEN1
SCHEMBL2487385 0.77 MAPT (0.66) MAPTRAB9ALMNANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 68 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108017060-B A kind of purification process of disilicone hexachloride 浙江博瑞电子科技有限公司 2019-06-28 CN claimed
CN-108017060-A A kind of purification process of disilicone hexachloride 浙江博瑞电子科技有限公司 2018-05-11 CN claimed
EP-2084163-B1 TETRACYCLIC INHIBITORS OF CYSTEINE PROTEASES, THE PHARMACEUTICAL COMPOSITIONS THEREOF AND THEIR THERAPEUTIC APPLICATIONS HYBRIGENICS SA (FR) 2017-04-12 EP claimed
US-8153791-B2 substituted pyrimidine compoundssuch as 4-amino-6-(3-chloro-4-fluoro-phenylamino)-pyrimidine-5-carbaldehyde O-methyl oxime, used for treating, preventing or ameliorating a chronic or acute protein kinase mediated diseasea, disorders or conditions JANSSEN PHARMACEUTICA N.V. (BE) 2012-04-10 US claimed
US-20070270425-A1 SUBSTITUTED PYRIMIDINYL OXIME KINASE INHIBITORS JANSSEN PHARMACEUTICA N.V. (BE) 2007-11-22 US claimed
EP-1075483-B1 HYGROMYCIN A DERIVATIVES PFIZER PROD INC (US) 2003-12-03 EP claimed
EP-1077984-B1 2\"-DEOXY HYGROMYCIN DERIVATIVES PFIZER PROD INC (US) 2003-06-18 EP claimed
US-6342497-B1 2″-deoxy hygromycin derivatives PFIZER INC 2002-01-29 US claimed
US-6313100-B1 ANTIBACTERIAL, ANTIPROTOZOA AGENTS PFIZER INC 2001-11-06 US claimed
EP-0445731-B1 Azabicyclo and azacyclo oxime and amine cholinergic agents and pharmaceutically acceptable salts thereof WARNER LAMBERT CO (US) 1996-01-10 EP claimed
US-5482938-A Azabicyclo and azacyclo oxime and amine cholinergic agents and methods of treatment WARNER-LAMBERT COMPANY (US) 1996-01-09 US claimed
EP-0138773-B1 USE OF QUINOLINE DERIVATIVES FOR THE PROTECTION OF CROP PLANTS CIBA-GEIGY AG (CH) 1990-08-29 EP claimed
US-4749406-A Quinoline derivatives and compositions thereof for the protection of cultivated plants CIBA-GEIGY CORPORATION (US) 1988-06-07 US claimed
US-4710508-A ANALGESICS WARNER-LAMBERT COMPANY (US) 1987-12-01 US claimed
EP-0138773-A2 Use of quinoline derivatives for the protection of crop plants CIBA-GEIGY AG (CH) 1985-04-24 EP claimed
CN-108017060-B A kind of purification process of disilicone hexachloride 浙江博瑞电子科技有限公司 2019-06-28 CN disclosed
CN-108017060-A A kind of purification process of disilicone hexachloride 浙江博瑞电子科技有限公司 2018-05-11 CN disclosed
US-4749406-A Quinoline derivatives and compositions thereof for the protection of cultivated plants CIBA-GEIGY CORPORATION (US) 1988-06-07 US disclosed
US-4710508-A ANALGESICS WARNER-LAMBERT COMPANY (US) 1987-12-01 US disclosed
EP-0138773-A2 Use of quinoline derivatives for the protection of crop plants CIBA-GEIGY AG (CH) 1985-04-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070270425-A1 SUBSTITUTED PYRIMIDINYL OXIME KINASE INHIBITORS MAP3K2, MAP3K1, MAP3K20 MAPT 3084/4885RAB9A 3964/4885LMNA 3862/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.