SCHEMBL5744486

SCHEMBL5744486

COCCN1C(=O)C(Nc2ccc(N3CCOCC3)cc2)=C(c2ccccc2)C1=O.COCCN1C(=O)C(Nc2ccc(SC)cc2)=C(c2ccccc2)C1=O.COCCN1C(=O)C(Nc2ccc3oc(C(C)=O)cc3c2)=C(c2ccccc2)C1=O.O=C1C(Nc2ccc(N3CCOCC3)cc2)=C(c2ccccc2)C(=O)N1Cc1cccnc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 3/20 0.37
NR1H3 Q13133 3/20 0.37
ACVR1 Q04771 3/20 0.36
NTRK1 P04629 1/20 0.35
HSD17B10 Q99714 3/20 0.35
ALDH1A1 P00352 3/20 0.35
KDM4E B2RXH2 2/20 0.35
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CASP1 P29466 2/20 0.34
HPGD P15428 1/20 0.34
ABCB1 P08183 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4692187 0.82 NR1H2 (0.47) NR1H2NR1H3HSD17B10ALDH1A1KDM4E
SCHEMBL4692190 0.79 NR1H2 (0.45) NR1H2NR1H3HSD17B10ALDH1A1KDM4E
SCHEMBL5747436 0.79 NR1H2 (0.44) NR1H2NR1H3HSD17B10ALDH1A1KDM4E
SCHEMBL4691823 0.78 NR1H2 (0.56) NR1H2NR1H3NTRK1ALDH1A1KDM4E
SCHEMBL5750387 0.76 NR1H2 (0.51) NR1H2NR1H3NTRK1ALDH1A1KDM4E
SCHEMBL4689410 0.75 NR1H2 (0.51) NR1H2NR1H3ACVR1HSD17B10ALDH1A1
SCHEMBL4688674 0.71 NR1H2 (0.56) NR1H2NR1H3MAPTSMN1; SMN2
SCHEMBL5737209 0.69 PTGS2 (0.49) NR1H2NR1H3ALDH1A1MAPTMEN1
SCHEMBL4690096 0.68 NR1H2 (0.51) NR1H2NR1H3NTRK1ALDH1A1KDM4E
SCHEMBL4688066 0.67 NR1H2 (0.80) NR1H2NR1H3ALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646626-A1 PYRROLE-2, 5-DIONE DERIVATIVES AS LIVER X RECEPTOR MODULATORS AstraZeneca AB (SE) 2006-04-19 EP claimed
WO-2005005417-A1 PYRROLE-2, 5-DIONE DERIVATIVES AS LIVER X RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2005-01-20 WO claimed