SCHEMBL5746178

SCHEMBL5746178

Cc1ccc(S(=O)(=O)N2CCC(c3ccc(Cl)cc3)CC2)cc1CC(=O)O

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
USP5 P45974 12/20 0.58
HDAC6 Q9UBN7 6/20 0.57
TP53 P04637 1/20 0.52
PTGDR2 Q9Y5Y4 3/20 0.49
USP3 Q9Y6I4 1/20 0.48
MAPT P10636 1/20 0.48
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
TSHR P16473 1/20 0.47
PTGDR Q13258 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5750977 0.91 PTGDR (0.50) USP5HDAC6PTGDR2MAPTKDM4E
SCHEMBL5749414 0.87 USP5 (0.52) USP5HDAC6TP53PTGDR2GAA
SCHEMBL5748257 0.83 PTGDR (0.56) HDAC6PTGDR2MAPTGAAPTGDR
SCHEMBL5749155 0.82 TSHR (0.47) USP5HDAC6PTGDR2MAPTKDM4E
SCHEMBL13804995 0.82 LSS (0.56) PTGDR2KDM4ELMNA
SCHEMBL5750800 0.81 USP5 (0.55) USP5HDAC6TP53PTGDR2USP3
SCHEMBL6353135 0.81 USP5 (0.57) USP5HDAC6TP53PTGDR2USP3
SCHEMBL13805201 0.80 CNR1 (0.58) GAALMNA
SCHEMBL13805065 0.79 KMT2A (0.60) PTGDR2LMNA
SCHEMBL13805135 0.78 MEN1 (0.53) PTGDR2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1735280-A1 ARYL SULFONAMIDE AND SULFONYL COMPOUNDS AS MODULATORS OF PPAR AND METHODS OF TREATING METABOLIC DISORDERS Kalypsys, Inc. (US) 2006-12-27 EP disclosed
WO-2005115983-A1 ARYL SULFONAMIDE AND SULFONYL COMPOUNDS AS MODULATORS OF PPAR AND METHODS OF TREATING METABOLIC DISORDERS KALYPSYS, INC. (US) 2005-12-08 WO disclosed
US-20050234046-A1 Aryl sulfonamide and sulfonyl compounds as modulators of PPAR and methods of treating metabolic disorders KALYPSYS, INC. (US) 2005-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050234046-A1 Aryl sulfonamide and sulfonyl compounds as modulators of PPAR and methods of treating metabolic disorders PPARA, PPARG, PPARD USP5 2874/4885HDAC6 838/4885TP53 2986/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.