SCHEMBL574695

SCHEMBL574695

CC(c1ccccc1)n1cc(C(N)=O)cn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 8/20 0.52
KLKB1 P03952 1/20 0.52
TDP1 Q9NUW8 2/20 0.42
ALDH1A1 P00352 1/20 0.42
ACHE P22303 2/20 0.42
PARP14 Q460N5 1/20 0.41
BRD4 O60885 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40
PARP1 P09874 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
HSD17B10 Q99714 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALKBH1 Q13686 1/20 0.40
LDHA P00338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL947911 0.88 CREBBP (0.55) CREBBPKLKB1TDP1ALDH1A1ACHE
SCHEMBL949676 0.88 CREBBP (0.55) CREBBPKLKB1TDP1ALDH1A1ACHE
SCHEMBL12913216 0.88 CREBBP (0.55) CREBBPKLKB1TDP1ALDH1A1ACHE
SCHEMBL949190 0.85 CREBBP (0.52) CREBBPKLKB1TDP1ALDH1A1ACHE
SCHEMBL947800 0.85 CREBBP (0.52) CREBBPKLKB1TDP1ALDH1A1ACHE
SCHEMBL949139 0.85 CREBBP (0.52) CREBBPKLKB1TDP1ALDH1A1ACHE
SCHEMBL20768103 0.82 KLKB1 (0.55) CREBBPKLKB1BRD4MAPTALKBH1
SCHEMBL28008347 0.81 KLKB1 (0.42) CREBBPKLKB1ALDH1A1ACHEPARP1
SCHEMBL30022092 0.81 TSHR (0.49) KLKB1ALDH1A1CYP3A4MAPTTSHR
SCHEMBL23212254 0.79 CYP1A2 (0.55) CREBBPKLKB1ALDH1A1CYP3A4MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112341390-B Compound for preparing targeted histone methyltransferase EZH2 covalent inhibitor and preparation method and application thereof 四川大学 2022-08-23 CN disclosed