SCHEMBL28008347

SCHEMBL28008347

Cc1ccccc1C(C)n1cc(C(N)=O)cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.42
OPRM1 P35372 1/20 0.42
OPRK1 P41145 1/20 0.42
KCNH2 Q12809 1/20 0.42
ACHE P22303 6/20 0.39
CHEK2 O96017 1/20 0.38
JAK1 P23458 1/20 0.36
TYK2 P29597 1/20 0.36
JAK3 P52333 1/20 0.36
ALDH1A1 P00352 1/20 0.36
USP1 O94782 1/20 0.35
WDR48 Q8TAF3 1/20 0.35
PARP1 P09874 1/20 0.35
PARP15 Q460N3 1/20 0.35
PARP10 Q53GL7 1/20 0.35
CREBBP Q92793 1/20 0.35
MEN1 O00255 1/20 0.35
PKM P14618 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL574695 0.81 CREBBP (0.52) KLKB1ACHEALDH1A1PARP1CREBBP
SCHEMBL659349 0.75 ACHE (0.64) ACHE
SCHEMBL28309802 0.74 ACHE (0.49) ACHEPARP10
SCHEMBL25819849 0.74 ACHE (0.49) ACHEPARP10
SCHEMBL12862846 0.72 ACHE (0.47) ACHE
SCHEMBL16323742 0.72 ALKBH2 (0.44) ACHEALDH1A1CREBBP
SCHEMBL25430220 0.71 ACHE (0.41) KLKB1ACHE
SCHEMBL20532460 0.71 CREBBP (0.71) CREBBP
SCHEMBL31322788 0.71 MAPK14 (0.49) ALDH1A1PARP1MEN1PKMKMT2A
SCHEMBL22399206 0.70 ACHE (0.68) ACHEJAK1TYK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103080104-B N-((6-amino-pyridin-3-yl)methyl)-heteroaryl-carboxamides as inhibitors of plasma kallikrein NOVARTIS AG 2015-04-08 CN disclosed