SCHEMBL5747489

SCHEMBL5747489

NC1CCN(c2ccc3c(C(=O)NCC4CCCCC4)cccc3n2)C1

nearest known ligand 0.49

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 7/20 0.49
ACACB O00763 6/20 0.46
ACACA Q13085 6/20 0.46
CNR1 P21554 4/20 0.44
CNR2 P34972 3/20 0.44
BCHE P06276 1/20 0.43
PRKCQ Q04759 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3837843 1.00 P2RX7 (0.49) P2RX7ACACBACACACNR1CNR2
SCHEMBL5747142 0.84 P2RX7 (0.54) P2RX7ACACBACACA
SCHEMBL1805331 0.84 P2RX7 (0.69) P2RX7
SCHEMBL1805240 0.84 P2RX7 (0.69) P2RX7
SCHEMBL1804304 0.84 P2RX7 (0.54) P2RX7ACACBACACA
SCHEMBL5767624 0.84 P2RX7 (0.69) P2RX7
Hydrochloric Acid SCHEMBL3842335 0.83 P2RX7 (0.68) P2RX7
SCHEMBL5745880 0.79 P2RX7 (0.67) P2RX7
SCHEMBL1803780 0.79 P2RX7 (0.67) P2RX7
SCHEMBL3837020 0.78 P2RX7 (0.65) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1633717-A1 NEW P2X7 RECEPTOR ANTAGONISTS AND THEIR USE AstraZeneca AB (SE) 2006-03-15 EP disclosed
WO-2004106305-A1 NEW P2X7 RECEPTOR ANTAGONISTS AND THEIR USE ASTRAZENECA AB (SE) 2004-12-09 WO disclosed