SCHEMBL5749544

SCHEMBL5749544

COc1ccc2ccc3ccc(N)c4ccc1c2c34

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.57
EP300 Q09472 1/20 0.55
KAT8 Q9H7Z6 1/20 0.55
ALDH1A1 P00352 8/20 0.45
CYP3A4 P08684 3/20 0.45
TDP1 Q9NUW8 3/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
ADRA2B P18089 1/20 0.43
PTGS1 P23219 1/20 0.43
NQO1 P15559 1/20 0.41
MAPT P10636 3/20 0.38
MEN1 O00255 2/20 0.38
THRB P10828 2/20 0.38
KMT2A Q03164 2/20 0.38
HTT P42858 2/20 0.38
GAA P10253 1/20 0.37
APP P05067 2/20 0.37
FGB P02675 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5746648 1.00 IDO1 (0.57) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL19999172 0.87 NQO1 (0.50) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL10392528 0.87 NQO1 (0.50) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL29876078 0.87 NQO1 (0.50) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL5746447 0.83 IDO1 (0.47) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL5746862 0.81 NQO1 (0.42) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL866016 0.80 KEAP1 (0.42) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL29372072 0.80 KEAP1 (0.42) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL867279 0.80 KEAP1 (0.42) IDO1EP300KAT8ALDH1A1CYP3A4
SCHEMBL2351815 0.79 HPGD (0.54) IDO1ALDH1A1CYP3A4TDP1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060293503-A1 Polyaminopyridines and method for producing same SUMITOMO SEIKA CHEMICALS CO., LTD (JP) 2006-12-28 US disclosed
EP-1669390-A1 POLYAMINOPYRIDINES AND METHOD FOR PRODUCING SAME SUMITOMO SEIKA CHEMICALS CO., LTD. (JP) 2006-06-14 EP disclosed