SCHEMBL5752686

SCHEMBL5752686

CC(C)(C)OC(=O)N1CCN(CCNC(=O)c2ccc(F)cc2)CC1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.60
DRD2 P14416 1/20 0.60
MAPK14 Q16539 1/20 0.59
ACKR3 P25106 1/20 0.58
CD274 Q9NZQ7 1/20 0.56
THRB P10828 1/20 0.54
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
HDAC2 Q92769 1/20 0.52
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
EPHX2 P34913 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4324960 0.90 CD274 (0.58) HTR1ADRD2MAPK14ACKR3CD274
SCHEMBL8404688 0.87 ACKR3 (0.57) MAPK14ACKR3CD274MEN1KMT2A
SCHEMBL8404689 0.86 ACKR3 (0.56) MAPK14ACKR3CD274MEN1KMT2A
SCHEMBL15947385 0.85 SMN1; SMN2 (0.59) MAPK14ACKR3CD274MEN1KMT2A
SCHEMBL31037305 0.85 DRD2 (0.58) DRD2MAPK14ACKR3CD274MEN1
SCHEMBL20458266 0.83 SMN1; SMN2 (0.56) MAPK14ACKR3CD274MEN1KMT2A
SCHEMBL18763563 0.82 MAPT (0.55) HTR1ADRD2MAPK14ACKR3MEN1
SCHEMBL31330228 0.81 ACKR3 (0.62) HTR1ADRD2ACKR3
SCHEMBL5749344 0.80 MEN1 (0.53) HTR1ADRD2ACKR3MEN1KMT2A
SCHEMBL19891463 0.79 DRD2 (0.59) DRD2ACKR3THRBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed