SCHEMBL5752817

SCHEMBL5752817

NC(Cc1ccc(C(F)(F)F)cc1)C(O)c1ccc(F)cc1F

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 3/20 0.49
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
TAAR1 Q96RJ0 1/20 0.38
CYP1A1 P04798 1/20 0.36
CYP1B1 Q16678 1/20 0.36
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
MAOB P27338 1/20 0.35
CHRM5 P08912 1/20 0.34
DPP4 P27487 2/20 0.34
MC4R P32245 1/20 0.34
IDO1 P14902 2/20 0.34
GRB2 P62993 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5752544 0.83 PDE2A (0.41) PDE2ATAAR1MAOBDPP4IDO1
SCHEMBL5752665 0.81 PDE2A (0.46) PDE2ACYP1A1CYP1B1CES2CES1
SCHEMBL6578585 0.80 TRPA1 (0.39) TAAR1CES2CES1IDO1GRB2
SCHEMBL5750053 0.80 TRPA1 (0.39) TAAR1CES2CES1IDO1GRB2
SCHEMBL5751727 0.80 TRPA1 (0.39) TAAR1CES2CES1IDO1GRB2
Hydrochloric Acid SCHEMBL5751082 0.79 TACR1 (0.39) TAAR1CES2CES1MAOBIDO1
SCHEMBL5753401 0.78 SLC7A5 (0.45) PDE2A
SCHEMBL5753231 0.77 PDE2A (0.40) PDE2ATAAR1CES2CES1MAOB
SCHEMBL5755207 0.73 PPARG (0.43) SLC6A2SLC6A4SLC6A3GRB2
SCHEMBL5750512 0.71 AKT1 (0.41) CYP3A4SLC6A2SLC6A4SLC6A3TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6982348-B2 Aminoethanol derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2006-01-03 US disclosed
US-20040127574-A1 Aminoethanol derivatives TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-07-01 US disclosed
EP-1362846-A1 AMINOETHANOL DERIVATIVES Takeda Chemical Industries, Ltd. (JP) 2003-11-19 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040127574-A1 Aminoethanol derivatives CETP, LCAT, MTTP PDE2A 2691/4885CYP3A4 775/4885CYP2D6 1951/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.