SCHEMBL5754867

SCHEMBL5754867

CC(C)C(C#N)(CCCN1CCN(CCOc2cccc(-c3ccccc3)c2)CC1)c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.54
CACNA1B Q00975 3/20 0.53
BACE1 P56817 1/20 0.53
HRH3 Q9Y5N1 7/20 0.50
MEN1 O00255 1/20 0.43
HTR1A P08908 1/20 0.43
HTR7 P34969 1/20 0.43
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
MAPK1 P28482 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
HTT P42858 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5750739 0.91 CACNA1B (0.48) LTA4HCACNA1BBACE1HRH3MEN1
SCHEMBL5752940 0.91 CACNA1B (0.48) LTA4HCACNA1BBACE1HRH3MEN1
SCHEMBL5754333 0.91 CACNA1B (0.58) LTA4HCACNA1BMEN1HTR1AKMT2A
SCHEMBL5753857 0.89 CACNA1B (0.54) CACNA1BMEN1KMT2A
SCHEMBL5752309 0.89 CACNA1B (0.52) LTA4HCACNA1BMEN1HTR1AHTR7
SCHEMBL5753351 0.89 CACNA1B (0.52) LTA4HCACNA1BMEN1HTR1AHTR7
SCHEMBL14432330 0.87 CACNA1B (0.53) CACNA1BHRH3MEN1KDM4EALDH1A1
SCHEMBL5753413 0.87 CACNA1B (0.58) CACNA1BMEN1
SCHEMBL5753739 0.85 CACNA1B (0.50) LTA4HCACNA1BHRH3MEN1KMT2A
SCHEMBL5752688 0.85 CACNA1B (0.49) LTA4HCACNA1BBACE1HRH3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP claimed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US claimed
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed