SCHEMBL5752940

SCHEMBL5752940

CC(C)C(C#N)(CCCN1CCN(CCOc2cccc(-c3ccsc3)c2)CC1)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.48
LTA4H P09960 1/20 0.44
BACE1 P56817 1/20 0.44
HRH3 Q9Y5N1 7/20 0.42
KDR P35968 1/20 0.41
MEN1 O00255 2/20 0.39
HRH2 P25021 1/20 0.38
HRH1 P35367 1/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
BMP4 P12644 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5754867 0.91 LTA4H (0.54) CACNA1BLTA4HBACE1HRH3MEN1
SCHEMBL5750739 0.85 CACNA1B (0.48) CACNA1BLTA4HBACE1HRH3MEN1
SCHEMBL5754333 0.84 CACNA1B (0.58) CACNA1BLTA4HMEN1HRH1KMT2A
SCHEMBL5753857 0.83 CACNA1B (0.54) CACNA1BMEN1HRH2HRH1KMT2A
SCHEMBL5753351 0.83 CACNA1B (0.52) CACNA1BLTA4HMEN1KMT2AKDM4E
SCHEMBL5752309 0.83 CACNA1B (0.52) CACNA1BLTA4HMEN1KMT2AKDM4E
SCHEMBL5238510 0.83 CACNA1B (0.45) CACNA1BHRH3MEN1KMT2AALDH1A1
SCHEMBL5241063 0.83 CACNA1B (0.47) CACNA1BHRH3MEN1HRH2HRH1
SCHEMBL14432330 0.81 CACNA1B (0.53) CACNA1BHRH3MEN1KMT2AKDM4E
SCHEMBL5241127 0.81 CACNA1B (0.46) CACNA1BHRH3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP claimed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US claimed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP claimed
EP-1099692-B1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES EISAI CO LTD (JP) 2006-05-03 EP disclosed
US-6737425-B1 SUCH AS 1-((4-CYANO-5-METHYL-4-PHENYL)HEXYL)-4-(2-(4-FLUORO -PHENOXY)ETHYL)PIPERAZINE; NERVE SELECTIVE CALCIUM ANTAGONISTS EISAI CO., LTD. (JP) 2004-05-18 US disclosed
EP-1099692-A1 N,N-SUBSTITUTED CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 2001-05-16 EP disclosed