SCHEMBL5755253

SCHEMBL5755253

COCCN(c1ccc(CNC(=O)c2ccc(C)n(-c3cccc(C(F)(F)F)c3)c2=O)cc1)S(C)(=O)=O

nearest known ligand 0.71

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ELANE P08246 16/20 0.71
CCR1 P32246 1/20 0.42
RECQL P46063 1/20 0.41
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5759763 0.92 ELANE (0.73) ELANECCR1
SCHEMBL5759599 0.91 ELANE (0.71) ELANECCR1
SCHEMBL5757514 0.90 ELANE (0.75) ELANECCR1
SCHEMBL5755626 0.90 ELANE (0.72) ELANECCR1
SCHEMBL5760864 0.89 ELANE (0.69) ELANECCR1
SCHEMBL5757023 0.88 ELANE (0.79) ELANECCR1RECQL
SCHEMBL5757012 0.87 ELANE (0.77) ELANECCR1
SCHEMBL5755005 0.85 ELANE (0.75) ELANECCR1
SCHEMBL5757397 0.84 ELANE (0.75) ELANECCR1RECQL
SCHEMBL5756976 0.83 ELANE (0.83) ELANECCR1RECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562902-B1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE ASTRAZENECA AB (SE) 2006-05-03 EP disclosed
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase ASRAZENECA AB (SE) 2006-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase SERPINB1, ELANE, SERPINE1 ELANE 2/4885CCR1 186/4885RECQL 107/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.