SCHEMBL5756294

SCHEMBL5756294

CN(C)CCCN(C(=O)c1ccc(Br)cc1)c1nc2cc(Cl)ccc2c(=O)n1Cc1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.70
CYP2C19 P33261 2/20 0.50
MAP1LC3B Q9GZQ8 1/20 0.50
CYP3A4 P08684 1/20 0.50
KCNH2 Q12809 1/20 0.50
GAA P10253 3/20 0.42
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
HTT P42858 1/20 0.41
MPO P05164 1/20 0.41
XDH P47989 1/20 0.41
CACNA1G O43497 2/20 0.41
KMT2A Q03164 2/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5760697 0.84 KIF11 (0.83) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2
Ck0106023 SCHEMBL12393608 0.82 KIF11 (1.00) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2
SCHEMBL1882393 0.81 KIF11 (0.65) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2
SCHEMBL1885255 0.81 KIF11 (0.64) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2
SCHEMBL12386697 0.80 KIF11 (0.79) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2
SCHEMBL12386717 0.79 KIF11 (0.78) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2
SCHEMBL1892039 0.79 KIF11 (0.78) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2
SCHEMBL14154542 0.79 KIF11 (0.91) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2
SCHEMBL1886208 0.78 KIF11 (0.61) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2
SCHEMBL5758646 0.76 KIF11 (0.72) KIF11CYP2C19MAP1LC3BCYP3A4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1689724-A1 QUINAZOLINONE COMPOUNDS AS ANTICANCER AGENTS Chiron Corporation (US) 2006-08-16 EP claimed
WO-2005051922-A1 QUINAZOLINONE COMPOUNDS AS ANTICANCER AGENTS CHIRON CORPORATION (US) 2005-06-09 WO claimed