SCHEMBL5757036

SCHEMBL5757036

COC(=O)N1CSC[C@H]1C(=O)NC(CNC(=O)c1ccccc1O)C(Cc1ccc(OC)cc1)SCC1CCCCC1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 3/20 0.45
ALDH1A1 P00352 2/20 0.35
PSMB8 P28062 7/20 0.34
P2RX7 Q99572 1/20 0.33
KMT2A Q03164 1/20 0.33
PSMB9 P28065 2/20 0.33
PSMB10 P40306 1/20 0.33
HSD17B10 Q99714 1/20 0.32
PSMB5 P28074 3/20 0.32
CTSS P25774 2/20 0.32
MMP9 P14780 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758645 0.95 CACNA1B (0.43) CACNA1BALDH1A1PSMB8P2RX7KMT2A
SCHEMBL5754912 0.95 CACNA1B (0.43) CACNA1BALDH1A1PSMB8P2RX7KMT2A
SCHEMBL5754438 0.95 CACNA1B (0.51) CACNA1BALDH1A1PSMB8HSD17B10CTSS
SCHEMBL5757099 0.94 CACNA1B (0.54) CACNA1BALDH1A1PSMB8P2RX7KMT2A
SCHEMBL5759035 0.89 CACNA1B (0.49) CACNA1BKMT2AHSD17B10
SCHEMBL5755981 0.88 KMT2A (0.38) CACNA1BALDH1A1P2RX7KMT2AHSD17B10
SCHEMBL5757463 0.88 CACNA1B (0.61) CACNA1BALDH1A1HSD17B10CTSS
SCHEMBL5758199 0.87 CACNA1B (0.43) CACNA1BPSMB8PSMB9PSMB10HSD17B10
SCHEMBL5754736 0.86 CACNA1B (0.40) CACNA1BKMT2AHSD17B10
SCHEMBL5752573 0.86 KDM4E (0.41) CACNA1BALDH1A1PSMB8P2RX7KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0997147-B1 AMINO ACID DERIVATIVES ONO PHARMACEUTICAL CO (JP) 2006-03-15 EP claimed