SCHEMBL5757077

SCHEMBL5757077

C(=C/c1nc(COc2ccc(CCCn3cccc3)cc2)co1)\c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 2/20 0.56
MINK1 Q8N4C8 1/20 0.56
FFAR1 O14842 3/20 0.43
ATP4A P20648 6/20 0.39
ATP4B P51164 6/20 0.39
HMOX1 P09601 1/20 0.38
HTT P42858 1/20 0.38
KMT2A Q03164 1/20 0.38
PPARG P37231 4/20 0.37
PPARA Q07869 4/20 0.37
CYSLTR2 Q9NS75 1/20 0.36
CYSLTR1 Q9Y271 1/20 0.36
LCK P06239 1/20 0.36
LTA4H P09960 1/20 0.36
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5757081 1.00 ERBB2 (0.56) ERBB2MINK1FFAR1ATP4AATP4B
SCHEMBL5755643 0.90 ERBB2 (0.54) ERBB2MINK1ATP4AATP4BHMOX1
SCHEMBL5755640 0.90 ERBB2 (0.54) ERBB2MINK1ATP4AATP4BHMOX1
SCHEMBL5790298 0.88 ERBB2 (0.60) ERBB2MINK1FFAR1ATP4AATP4B
SCHEMBL5790299 0.88 ERBB2 (0.60) ERBB2MINK1FFAR1ATP4AATP4B
SCHEMBL5759021 0.88 ERBB2 (0.55) ERBB2MINK1FFAR1ATP4AATP4B
SCHEMBL5759019 0.88 ERBB2 (0.55) ERBB2MINK1FFAR1ATP4AATP4B
SCHEMBL5760882 0.88 ERBB2 (0.57) ERBB2MINK1ATP4AATP4BHMOX1
SCHEMBL5760885 0.88 ERBB2 (0.57) ERBB2MINK1ATP4AATP4BHMOX1
SCHEMBL5761163 0.87 ERBB2 (0.57) ERBB2MINK1ATP4AATP4BHMOX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed