SCHEMBL5790299

SCHEMBL5790299

C(=Cc1nc(COc2ccc(CCCn3cccn3)cc2)co1)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERBB2 P04626 2/20 0.60
MINK1 Q8N4C8 1/20 0.60
FFAR1 O14842 3/20 0.40
TP53 P04637 2/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HMOX1 P09601 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
ATP4A P20648 5/20 0.35
ATP4B P51164 5/20 0.35
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
CYSLTR2 Q9NS75 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5790298 1.00 ERBB2 (0.60) ERBB2MINK1FFAR1TP53MAPT
SCHEMBL26316546 0.89 ERBB2 (0.63) ERBB2MINK1FFAR1MAPTNPC1
SCHEMBL5759321 0.89 ERBB2 (0.75) ERBB2MINK1FFAR1MAPTHMOX1
SCHEMBL5759315 0.89 ERBB2 (0.75) ERBB2MINK1FFAR1MAPTHMOX1
SCHEMBL5759019 0.88 ERBB2 (0.55) ERBB2MINK1FFAR1HTTKMT2A
SCHEMBL5759021 0.88 ERBB2 (0.55) ERBB2MINK1FFAR1HTTKMT2A
SCHEMBL5757081 0.88 ERBB2 (0.56) ERBB2MINK1FFAR1HMOX1HTT
SCHEMBL5757077 0.88 ERBB2 (0.56) ERBB2MINK1FFAR1HMOX1HTT
SCHEMBL780445 0.88 ERBB2 (0.55) ERBB2MINK1FFAR1TP53MAPT
SCHEMBL780446 0.88 ERBB2 (0.55) ERBB2MINK1FFAR1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed