SCHEMBL5757095

SCHEMBL5757095

O=C(c1ccccc1)C1CCN(CCCN(c2ccccc2)S(=O)(=O)c2ccccc2[N+](=O)[O-])CC1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
TDP1 Q9NUW8 1/20 0.50
HTR2A P28223 3/20 0.48
KCNH2 Q12809 2/20 0.47
ALDH1A1 P00352 3/20 0.46
MAPT P10636 2/20 0.46
CYP2D6 P10635 3/20 0.44
NPSR1 Q6W5P4 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP2C9 P11712 1/20 0.44
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
KDM4E B2RXH2 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5756938 0.94 HTR2A (0.52) KMT2ATDP1HTR2ACYP2D6KDM4E
SCHEMBL5757056 0.83 KCNH2 (0.56) HTR2AKCNH2CYP2D6KDM4ECYP1A2
SCHEMBL5754009 0.83 KMT2A (0.49) KMT2ATDP1ALDH1A1MAPTMEN1
SCHEMBL12311334 0.74 KMT2A (0.54) KMT2ATDP1ALDH1A1MAPTCYP2D6
SCHEMBL16975882 0.74 NPSR1 (0.56) KMT2ATDP1ALDH1A1MAPTCYP2D6
SCHEMBL5758878 0.74 GRIN2B (0.50) KMT2AHTR2AALDH1A1MAPTCYP2D6
SCHEMBL6008687 0.73 HTR2A (0.47) KMT2AHTR2AKCNH2ALDH1A1MAPT
SCHEMBL5754844 0.72 KCNH2 (0.60) HTR2AKCNH2CYP2D6KDM4ECYP1A2
SCHEMBL5758044 0.71 KCNH2 (0.62) HTR2AKCNH2CYP2D6KDM4ECYP1A2
SCHEMBL4395372 0.71 KMT2A (0.55) KMT2ATDP1HTR2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401821-A4 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORP (KR) 2006-05-31 EP claimed
EP-1401821-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK Corporation (KR) 2004-03-31 EP claimed
WO-2002100848-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORPORATION (KR) 2002-12-19 WO claimed
EP-1401821-A4 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORP (KR) 2006-05-31 EP disclosed
EP-1401821-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK Corporation (KR) 2004-03-31 EP disclosed
WO-2002100848-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORPORATION (KR) 2002-12-19 WO disclosed