SCHEMBL5754844

SCHEMBL5754844

O=C(c1ccccc1)C1CCN(CCCN(C(=O)c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.60
PTGIR P43119 4/20 0.58
HTR2A P28223 2/20 0.57
ACHE P22303 1/20 0.55
CCR5 P51681 1/20 0.53
ADRA2C P18825 1/20 0.52
KDM4E B2RXH2 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
HRH3 Q9Y5N1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5758647 0.83 CCR5 (0.67) PTGIRACHECCR5
SCHEMBL5758121 0.83 ADRA2C (0.61) PTGIRHTR2AACHEADRA2CKDM4E
SCHEMBL28602611 0.82 KCNH2 (0.64) KCNH2ACHECCR5
SCHEMBL5758044 0.82 KCNH2 (0.62) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL5758945 0.81 KCNH2 (0.54) KCNH2HTR2ACCR5
SCHEMBL8710869 0.80 ACHE (0.56) PTGIRHTR2AACHEKDM4ECYP1A2
SCHEMBL5757056 0.79 KCNH2 (0.56) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL7250766 0.79 KCNH2 (0.72) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL8313722 0.78 KCNH2 (0.71) KCNH2HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL8664405 0.77 PTGIR (0.50) KCNH2PTGIRHTR2AACHEHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401821-A4 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORP (KR) 2006-05-31 EP claimed
EP-1401821-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK Corporation (KR) 2004-03-31 EP claimed
WO-2002100848-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORPORATION (KR) 2002-12-19 WO claimed
EP-1401821-A4 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORP (KR) 2006-05-31 EP disclosed
EP-1401821-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK Corporation (KR) 2004-03-31 EP disclosed
WO-2002100848-A1 NOVEL PHENYLALKYL DIAMINE AND AMIDE ANALOGS SK CORPORATION (KR) 2002-12-19 WO disclosed