SCHEMBL5757500

SCHEMBL5757500

Cc1ccc(C(=O)NOc2ccccc2)c(=O)n1-c1cccc(C(F)(F)F)c1

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.58
NOTUM Q6P988 1/20 0.50
PLA2G10 O15496 1/20 0.43
CYP1A2 P05177 1/20 0.43
GSR P00390 3/20 0.43
TP53 P04637 2/20 0.43
MAPT P10636 2/20 0.43
POLB P06746 1/20 0.42
NPY5R Q15761 3/20 0.41
PPARG P37231 1/20 0.40
PTGER1 P34995 1/20 0.40
FAAH O00519 1/20 0.40
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5756494 0.88 ELANE (0.73) ELANENOTUM
SCHEMBL31490303 0.84 ELANE (0.48) ELANENOTUMPLA2G10CYP1A2GSR
SCHEMBL560944 0.84 ELANE (0.48) ELANENOTUMPLA2G10CYP1A2GSR
SCHEMBL5445143 0.83 PLA2G10 (0.56) ELANENOTUMPLA2G10CYP1A2GSR
SCHEMBL5759984 0.82 ELANE (0.73) ELANETP53PPARG
SCHEMBL11895153 0.82 NOTUM (0.47) ELANENOTUMPLA2G10CYP1A2GSR
SCHEMBL5755788 0.82 ELANE (0.79) ELANENOTUMMAPTPOLBLMNA
SCHEMBL5757787 0.82 ELANE (0.59) ELANENOTUMMAPTPOLBNPY5R
SCHEMBL561046 0.82 NOTUM (0.68) ELANENOTUMCYP1A2GSRMAPT
SCHEMBL5758541 0.81 ELANE (0.59) ELANENOTUMPLA2G10CYP1A2GSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562902-B1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE ASTRAZENECA AB (SE) 2006-05-03 EP disclosed
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase ASRAZENECA AB (SE) 2006-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase SERPINB1, ELANE, SERPINE1 ELANE 2/4885NOTUM 3748/4885PLA2G10 312/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.