SCHEMBL5759566

SCHEMBL5759566

Cc1ccc(C(=O)NC(C)c2ccc(F)cc2)c(=O)n1-c1cccc(C#N)c1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 9/20 0.45
CNR1 P21554 5/20 0.45
NOTUM Q6P988 1/20 0.44
PTGDR2 Q9Y5Y4 1/20 0.43
KCNK3 O14649 1/20 0.41
PTGER4 P35408 2/20 0.41
PDE10A Q9Y233 2/20 0.40
PDPK1 O15530 1/20 0.40
PTGER2 P43116 1/20 0.40
LIPG Q9Y5X9 1/20 0.40
GPR139 Q6DWJ6 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5756499 0.91 CNR1 (0.54) CNR2CNR1NOTUMPTGER4PTGER2
SCHEMBL5759245 0.90 PTGER4 (0.45) CNR2CNR1NOTUMPTGER4PTGER2
SCHEMBL5755823 0.82 ELANE (0.58) NOTUMLIPG
SCHEMBL5757117 0.80 ELANE (0.47) CNR2CNR1NOTUM
SCHEMBL5755952 0.77 ELANE (0.47) NOTUMPDE10A
SCHEMBL5930971 0.76 NOTUM (0.43) CNR2CNR1NOTUM
SCHEMBL5757706 0.76 ELANE (0.45) CNR2CNR1NOTUM
SCHEMBL5756492 0.75 ELANE (0.57) CNR2CNR1NOTUMPTGER4LIPG
SCHEMBL5756526 0.75 ELANE (0.57) CNR2CNR1NOTUMPTGER4LIPG
SCHEMBL5757651 0.75 ELANE (0.54) CNR2CNR1NOTUMPTGER4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562902-B1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE ASTRAZENECA AB (SE) 2006-05-03 EP disclosed
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase ASRAZENECA AB (SE) 2006-02-16 US disclosed
CN-1711243-A 2-pyridone derivatives as inhibitors of neutrophil elastase ASTRAZENECA AB (SE) 2005-12-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase SERPINB1, ELANE, SERPINE1 CNR2 2164/4885CNR1 2232/4885NOTUM 3748/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.