SCHEMBL5760458

SCHEMBL5760458

CCCCCC(=O)CNCc1cc(-c2ccc(CCC(=O)OOCC)cc2)cs1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C8 P10632 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2B6 P20813 1/20 0.35
CYP2C19 P33261 1/20 0.35
RARB P10826 9/20 0.33
AVPR1B P47901 1/20 0.33
RARA P10276 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
MTOR P42345 1/20 0.33
KMT2A Q03164 1/20 0.33
S1PR1 P21453 3/20 0.32
S1PR3 Q99500 3/20 0.32
S1PR2 O95136 2/20 0.32
TRPV1 Q8NER1 1/20 0.32
LPAR2 Q9HBW0 1/20 0.32
IAPP P10997 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5761809 0.84 CYP4F2 (0.36) CYP4F2CYP4A11
SCHEMBL5760450 0.82 KMT2A (0.35) RARBRARAMEN1ALDH1A1MAPT
SCHEMBL1750019 0.78 PTPRF (0.41)
SCHEMBL2217322 0.78 PTPRF (0.41)
SCHEMBL2220220 0.75 MME (0.41) ALDH1A1
SCHEMBL5761770 0.73 PTPRF (0.36)
SCHEMBL67799 0.71 CYP4F2 (0.43) RARBRARAMEN1ALDH1A1MAPT
SCHEMBL68143 0.71 RARB (0.38) RARBRARAS1PR1S1PR3S1PR2
SCHEMBL1749562 0.71 PPARA (0.43)
SCHEMBL1750609 0.70 HDAC1 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638964-A1 NOVEL COMPOUNDS THAT MODULATE PPAR-GAMMA TYPE RECEPTORS, AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS Galderma Research & Development, S.N.C. (FR) 2006-03-29 EP disclosed
WO-2004113331-A1 NOVEL COMPOUNDS THAT MODULATE PPARϜ TYPE RECEPTORS, AND USE THEREOF IN COSMETIC OR PHARMACEUTICAL COMPOSITIONS GALDERMA RESEARCH & DEVELOPMENT, S.N.C. (FR) 2004-12-29 WO disclosed