SCHEMBL5761752

SCHEMBL5761752

CN(C(=O)C1CCN(C(=O)OCc2ccccc2)CC1)C(c1ccnc(F)c1)C(O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
CYP2C19 P33261 1/20 0.41
HTT P42858 1/20 0.40
GRIN2B Q13224 9/20 0.38
FAAH O00519 1/20 0.38
TRPV4 Q9HBA0 1/20 0.38
LNPEP Q9UIQ6 1/20 0.38
OPRK1 P41145 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM3 P20309 1/20 0.37
F2R P25116 1/20 0.37
TACR1 P25103 1/20 0.36
CYP2D6 P10635 3/20 0.36
CYP2C9 P11712 3/20 0.36
CYP3A4 P08684 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6280979 0.88 GRIN2B (0.42) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL6189868 0.79 SMN1; SMN2 (0.44) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL6280976 0.79 SMN1; SMN2 (0.41) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL7994460 0.78 FOLH1 (0.37) HTTOPRK1
SCHEMBL7679543 0.77 SMN1; SMN2 (0.43) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL7467972 0.71 SMN1; SMN2 (0.41) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL7672577 0.70 SMN1; SMN2 (0.46) SMN1; SMN2NPC1RAB9ACYP2C19HTT
SCHEMBL7469105 0.69 TRPC3 (0.44) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL4025102 0.69 MAPK14 (0.52) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B
SCHEMBL8011517 0.69 MAPK14 (0.52) SMN1; SMN2NPC1RAB9ACYP2C19GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1414443-B1 BENZIMIDAZO 4,5-f|ISOQUINOLINONE DERIVATIVES MERCK & CO INC (US) 2006-11-15 EP disclosed