SCHEMBL5762013

SCHEMBL5762013

CN(c1ncc(Br)cn1)S(C)(=O)=O.[NaH]

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 1/20 0.33
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 1/20 0.31
ALOX15 P16050 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP19A1 P11511 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2113176 0.98 EDNRA (0.34) EDNRAKDM4EALDH1A1ALOX15HSD17B10
SCHEMBL5762009 0.94 EDNRA (0.33) EDNRA
SCHEMBL19782813 0.78 CA12 (0.35) KDM4EALDH1A1ALOX15HSD17B10CYP19A1
SCHEMBL1751661 0.76 KMT2A (0.39) ALDH1A1ALOX15HSD17B10
SCHEMBL567737 0.73 CYP19A1 (0.33) CYP19A1
SCHEMBL2067485 0.72 PIK3C3 (0.45) EDNRAHSD17B10CYP19A1
SCHEMBL3132631 0.72 KDM4E (0.43) KDM4EALDH1A1ALOX15HSD17B10
SCHEMBL629463 0.71 ALDH1A1 (0.48) EDNRAKDM4EALDH1A1ALOX15HSD17B10
SCHEMBL28940994 0.69 KMT2A (0.35) KDM4EALDH1A1ALOX15HSD17B10
SCHEMBL28940996 0.69 HDAC1 (0.40) KDM4EALDH1A1ALOX15HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611091-A1 NOVEL COMPOUNDS AstraZeneca AB (SE) 2006-01-04 EP disclosed
WO-2004089885-A1 NOVEL COMPOUNDS ASTRAZENECA AB (SE) 2004-10-21 WO disclosed