SCHEMBL5763148

SCHEMBL5763148

CC(C)(C)[Si](C)(C)OC(CNCCCCCNC(=O)O)c1ccc(OCc2ccccc2)c2[nH]c(=O)ccc12

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 17/20 0.42
ADRB1 P08588 13/20 0.42
DRD2 P14416 2/20 0.40
DRD1 P21728 2/20 0.40
DRD4 P21917 2/20 0.40
DRD3 P35462 2/20 0.40
KDM4E B2RXH2 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5763122 1.00 ADRB2 (0.42) ADRB2ADRB1DRD2DRD1DRD4
SCHEMBL17633021 1.00 ADRB2 (0.42) ADRB2ADRB1DRD2DRD1DRD4
SCHEMBL28423974 0.98 ADRB2 (0.42) ADRB2ADRB1DRD2DRD1DRD4
SCHEMBL28423971 0.98 ADRB2 (0.42) ADRB2ADRB1DRD2DRD1DRD4
SCHEMBL963630 0.93 ADRB2 (0.42) ADRB2ADRB1DRD2DRD1DRD4
SCHEMBL963632 0.93 ADRB2 (0.42) ADRB2ADRB1DRD2DRD1DRD4
SCHEMBL963633 0.93 ADRB2 (0.42) ADRB2ADRB1DRD2DRD1DRD4
SCHEMBL18259968 0.92 ADRB2 (0.44) ADRB2ADRB1DRD2DRD1DRD4
SCHEMBL18259967 0.92 ADRB2 (0.44) ADRB2ADRB1DRD2DRD1DRD4
SCHEMBL28423946 0.91 ADRB2 (0.42) ADRB2ADRB1DRD2DRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1615881-A2 DIARYLMETHYL AND RELATED COMPOUNDS HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY Theravance, Inc. (US) 2006-01-18 EP disclosed
WO-2004089892-A2 DIARYLMETHYL AND RELATED COMPOUNDS HAVING BETA2 ANDRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY THERAVANCE, INC. (US) 2004-10-21 WO disclosed